Compile Data Set for Download or QSAR
Found 360 with Last Name = 'caldwell' and Initial = 'jj'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307954(4-((4-Chlorobenzyloxy)methyl)-1-(7H-pyrrolo[2,3-d]...)copy SMILEScopy InChI
Affinity DataIC50: 0.590nMAssay Description:Inhibition of PKB in human U87MG cells assessed as GSK3beta phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50237622(4-(4-Chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-4...)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMAssay Description:Inhibition of PKB in human U87MG cells assessed as GSK3beta phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307955(4-(2,4-Dichlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimid...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PKB in human PC3M cells assessed as GSK3beta phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307942(4-Amino-N-(4-chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376061(CHEMBL409503)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335684(4-FLUORO-2-(4-{[(3S,4R)-4-(1-HYDROXY-1-METHYLETHYL...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50237622(4-(4-Chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-4...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PKB in human PC3M cells assessed as GSK3beta phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307956(4-Amino-N-(2,4-dichlorobenzyl)-1-(7H-pyrrolo[2,3-d...)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibition of PKB in human PC3M cells assessed as GSK3beta phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307957(4-Amino-N-(4-chloro-2-fluorobenzyl)-1-(7H-pyrrolo[...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307975(4-Amino-N-(4-chlorobenzyl)-N-methyl-1-(7H-pyrrolo[...)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of PKB in human PC3M cells assessed as GSK3beta phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307956(4-Amino-N-(2,4-dichlorobenzyl)-1-(7H-pyrrolo[2,3-d...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376067(CHEMBL260000)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335683(4-fluoro-2-(4-((3S,4R)-4-(2-hydroxypropan-2-yl)pyr...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RHXPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307958(4-Amino-N-(4-chlorobenzyl)-1-(8-oxo-8,9-dihydro-7H...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307959(4-(4-Chlorobenzyl)-1-(1H-pyrrolo[2,3-b]pyridin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307960(4-Amino-N-(3,4-dichlorobenzyl)-1-(7H-pyrrolo[2,3-d...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50237622(4-(4-Chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-4...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50237622(4-(4-Chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-4...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307945(4-(4-tert-Butylbenzyl)-1-(1H-pyrazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibition of PKB in human U87MG cells assessed as GSK3beta phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376060(CHEMBL407504)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307961(4-(Naphthalen-2-ylmethyl)-1-(7H-pyrrolo[2,3-d]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307962(4-Amino-N-(3-chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376059(CHEMBL259998)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307966(4-Amino-N-(4-chlorobenzyl)-1-(1H-pyrrolo[2,3-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Inhibition of PKB in human U87MG cells assessed as GSK3beta phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335687(2-(4-((3S,4R)-4-(2-hydroxypropan-2-yl)pyrrolidin-3...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RHXPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376063(CHEMBL406863)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307954(4-((4-Chlorobenzyloxy)methyl)-1-(7H-pyrrolo[2,3-d]...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307963(4-Amino-N-(2-chloro-4-fluorobenzyl)-1-(7H-pyrrolo[...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307955(4-(2,4-Dichlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimid...)copy SMILEScopy InChI
Affinity DataIC50: 8.5nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335662((S)-4-(1H-pyrazol-3-yl)-2-(4-(pyrrolidin-3-ylamino...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RHXPubMedMMDB
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307964(4-Amino-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-N-(4-(...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307965(4-Amino-N-(2,4-difluorobenzyl)-1-(7H-pyrrolo[2,3-d...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335685(4-fluoro-2-(4-((3S,4R)-4-(hydroxymethyl)pyrrolidin...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RHXPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335681((S)-4-fluoro-2-(7-(2-methoxyethoxy)-4-(pyrrolidin-...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RHXPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307966(4-Amino-N-(4-chlorobenzyl)-1-(1H-pyrrolo[2,3-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307967(4-(4-Chlorobenzyl)-1-(1H-pyrazolo[3,4-b]pyridin-4-...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335680((S)-2-(6,7-dimethoxy-4-(pyrrolidin-3-ylamino)quina...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RHXPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376064(CHEMBL260577)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335686(2-(4-((3S,4R)-4-(2-hydroxypropan-2-yl)pyrrolidin-3...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RHXPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307968(4-Amino-N-(4-fluorobenzyl)-1-(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307969(4-(3-Methoxybenzyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307970(4-(2,5-Dichlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimid...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376068(CHEMBL260358)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307971(4-(3,4-Dichlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimid...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307972(4-(3-(Trifluoromethoxy)benzyl)-1-(7H-pyrrolo[2,3-d...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50307973(4-(2,6-Dichlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimid...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of PKBbeta by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B608VPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM16232(6-phenylpurine compound 20 | 6-{4-[4-(4-chlorophen...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50335671(4-fluoro-2-(4-((3S,4R)-4-(2-hydroxypropan-2-yl)pyr...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of CHK2 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RHXPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376062(CHEMBL260463)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50376058(CHEMBL259999)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of PKBbeta recombinant by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63NV8PubMed
Displayed 1 to 50 (of 360 total ) | Next | Last >>
Jump to: