Compile Data Set for Download or QSAR
Found 514 with Last Name = 'mills' and Initial = 'jj'
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605348(CHEMBL5183319)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468736(US10807959, Example 5)copy SMILEScopy InChI
Affinity DataKi:  0.0200nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605350(CHEMBL5177656)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605349(CHEMBL5191181)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605347(CHEMBL5174178)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605346(CHEMBL5177738)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605343(CHEMBL5190556)copy SMILES
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605336(CHEMBL5202831)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605332(CHEMBL5195031)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605331(CHEMBL5190578)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605330(CHEMBL5201192)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605325(CHEMBL5199203)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605352(CHEMBL5198319)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605353(CHEMBL5190717)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605350(CHEMBL5177656)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605355(CHEMBL5170717)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605356(CHEMBL5170071)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50520131(CHEMBL4588661)copy SMILEScopy InChI
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605323(CHEMBL5174357)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468925(US10807959, Example B64)copy SMILEScopy InChI
Affinity DataKi:  0.0210nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605322(CHEMBL5169425)copy SMILES
Affinity DataKi:  0.0220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605327(CHEMBL5181314)copy SMILES
Affinity DataKi:  0.0230nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605329(CHEMBL5186072)copy SMILES
Affinity DataKi:  0.0250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605339(CHEMBL5171051)copy SMILES
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605354(CHEMBL5179388)copy SMILES
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605337(CHEMBL5192283)copy SMILES
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605351(CHEMBL5180435)copy SMILES
Affinity DataKi:  0.0290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605324(CHEMBL5182982)copy SMILES
Affinity DataKi:  0.0290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50521464(CHEMBL4469869 | US11596639, Example 78)copy SMILEScopy InChI
Affinity DataKi:  0.0300nMAssay Description:Inhibition of FITC-labeled Bak peptide binding to MBP-fused Mcl-1 (unknown origin) measured after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50521464(CHEMBL4469869 | US11596639, Example 78)copy SMILEScopy InChI
Affinity DataKi:  0.0300nMAssay Description:Inhibition of FITC-labeled Bak peptide binding to MBP-fused Mcl-1 (unknown origin) measured after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50521464(CHEMBL4469869 | US11596639, Example 78)copy SMILEScopy InChI
Affinity DataKi:  0.0300nMAssay Description:Inhibition of FITC-labeled Bak peptide binding to MBP-fused Mcl-1 (unknown origin) measured after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468927(US10807959, Example B74)copy SMILEScopy InChI
Affinity DataKi:  0.0310nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468928(US10807959, Example B81)copy SMILEScopy InChI
Affinity DataKi:  0.0330nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605318(CHEMBL5171315)copy SMILES
Affinity DataKi:  0.0330nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605319(CHEMBL5171953)copy SMILES
Affinity DataKi:  0.0350nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605320(CHEMBL5202878)copy SMILES
Affinity DataKi:  0.0360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468938(US10807959, Example B109)copy SMILEScopy InChI
Affinity DataKi:  0.0380nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605342(CHEMBL5194215)copy SMILES
Affinity DataKi:  0.0390nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50520121(CHEMBL4441671 | US10844044, Example 1)copy SMILEScopy InChI
Affinity DataKi:  0.0440nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605326(CHEMBL5206455)copy SMILES
Affinity DataKi:  0.0460nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605321(CHEMBL5182077)copy SMILES
Affinity DataKi:  0.0550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605345(CHEMBL5190202)copy SMILES
Affinity DataKi:  0.0640nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50521465(CHEMBL4449014 | US11596639, Example 88)copy SMILEScopy InChI
Affinity DataKi:  0.0810nMAssay Description:Inhibition of FITC-labeled Bak peptide binding to MBP-fused Mcl-1 (unknown origin) measured after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69P04PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468936(US10807959, Example B99)copy SMILEScopy InChI
Affinity DataKi:  0.0870nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468939(US10807959, Example B111)copy SMILEScopy InChI
Affinity DataKi:  0.0870nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468945(US10807959, Example B129)copy SMILEScopy InChI
Affinity DataKi:  0.0890nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468937(US10807959, Example B107)copy SMILEScopy InChI
Affinity DataKi:  0.0970nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468816(US10807959, Example 86)copy SMILEScopy InChI
Affinity DataKi: <0.100nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468797(US10807959, Example 67)copy SMILEScopy InChI
Affinity DataKi: <0.100nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM468835(US10807959, Example 105)copy SMILEScopy InChI
Affinity DataKi: <0.100nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q219XUS Patent
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