Compile Data Set for Download or QSAR
Found 25 with Last Name = 'qin' and Initial = 'jj'
LigandPNGBDBM50408828(CHEMBL5270588)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408825(CHEMBL5280147)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
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LigandPNGBDBM50408825(CHEMBL5280147)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408825(CHEMBL5280147)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408825(CHEMBL5280147)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408829(CHEMBL5278293)copy SMILEScopy InChI
Affinity DataIC50: 3.57E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50446146(CHEMBL3108909)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50446146(CHEMBL3108909)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99MKPubMed
LigandPNGBDBM50605550(C-188-9 | Stat3 inhibitor c188-9 | Stat3 inhibitor...)copy SMILES
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50446145(CHEMBL3108910)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50446145(CHEMBL3108910)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99MKPubMed
LigandPNGBDBM50353432(CHEMBL1829876 | US10196373, Compound 45O)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50353432(CHEMBL1829876 | US10196373, Compound 45O)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99MKPubMed
LigandPNGBDBM50408835(CHEMBL5267904)copy SMILEScopy InChI
Affinity DataIC50: 7.50E+3nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
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LigandPNGBDBM50408832(CHEMBL4168135)copy SMILEScopy InChI
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408834(CHEMBL5271424)copy SMILEScopy InChI
Affinity DataIC50: 5.08E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM20283(2-hydroxy-4-(2-{[(4-methylbenzene)sulfonyl]oxy}ace...)copy SMILEScopy InChI
Affinity DataIC50: 8.60E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99MKPubMed
LigandPNGBDBM50408834(CHEMBL5271424)copy SMILEScopy InChI
Affinity DataIC50: 1.13E+5nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408833(CHEMBL5277569)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408831(CHEMBL5271534)copy SMILEScopy InChI
Affinity DataKd:  6.60E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408827(CHEMBL5282950)copy SMILEScopy InChI
Affinity DataKd:  1.55E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408830(CHEMBL5284089)copy SMILEScopy InChI
Affinity DataKd:  3.30E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50353432(CHEMBL1829876 | US10196373, Compound 45O)copy SMILEScopy InChI
Affinity DataKd:  504nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408826(CHEMBL5268863)copy SMILEScopy InChI
Affinity DataKd:  4.50E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408830(CHEMBL5284089)copy SMILEScopy InChI
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails