Compile Data Set for Download or QSAR
Found 282 with Last Name = 'terebetski' and Initial = 'jl'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021345(CHEMBL3287928)copy SMILEScopy InChI
Affinity DataKi:  637nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12KNPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021331(CHEMBL3287930)copy SMILEScopy InChI
Affinity DataKi:  740nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12KNPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350538(CHEMBL1812717)copy SMILEScopy InChI
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12KNPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021346(CHEMBL3287926)copy SMILEScopy InChI
Affinity DataKi:  1.54E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12KNPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021329(CHEMBL3287932)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12KNPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021344(CHEMBL3287929)copy SMILEScopy InChI
Affinity DataKi:  5.21E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12KNPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021334(CHEMBL3287931)copy SMILEScopy InChI
Affinity DataKi:  2.85E+4nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12KNPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021330(CHEMBL3287927)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12KNPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362418(CHEMBL1938418)copy SMILEScopy InChI
Affinity DataIC50: 0.180nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362419(CHEMBL1940544)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434318(CHEMBL2386566)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362420(CHEMBL1940540)copy SMILEScopy InChI
Affinity DataIC50: 0.330nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434329(CHEMBL2386554)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362417(CHEMBL1940545)copy SMILEScopy InChI
Affinity DataIC50: 0.420nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)copy SMILEScopy InChI
Affinity DataIC50: 0.430nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434329(CHEMBL2386554)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434316(CHEMBL2386568)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434318(CHEMBL2386566)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362417(CHEMBL1940545)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)copy SMILEScopy InChI
Affinity DataIC50: 0.690nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434317(CHEMBL2386567)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362419(CHEMBL1940544)copy SMILEScopy InChI
Affinity DataIC50: 0.860nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434315(CHEMBL2386569)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434313(CHEMBL2386571)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434314(CHEMBL2386570)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434322(CHEMBL2386562)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362418(CHEMBL1938418)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434314(CHEMBL2386570)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434316(CHEMBL2386568)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434315(CHEMBL2386569)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434320(CHEMBL2386564)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434313(CHEMBL2386571)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434317(CHEMBL2386567)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362420(CHEMBL1940540)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362415(CHEMBL1940536)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362411(CHEMBL1940541)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362413(CHEMBL1940538)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362410(CHEMBL1940542)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362437(CHEMBL1940367)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434319(CHEMBL2386565)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434319(CHEMBL2386565)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362430(CHEMBL1940526)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434321(CHEMBL2386563)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434323(CHEMBL2386561)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434320(CHEMBL2386564)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434328(CHEMBL2386555)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6RWJPubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84CB4PubMed
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