TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 9.70nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 83nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 157nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: 277nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Vanderbilt University Institute of Imaging Science (VUIIS)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Displacement of [3H] substance P from recombinant human NK1 receptor expressed in CHO cells after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate preincubated for 15 mins followed by NADPH addition measured after 8 min...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Negative allosteric modulation of rat mGlu7 receptor expressed in HEK cells co-expressing Galphai5 assessed as decrease in glutamate-induced thallium...More data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate preincubated for 15 mins followed by NADPH addition measured after 8 min...More data for this Ligand-Target Pair