Compile Data Set for Download or QSAR
Found 201 with Last Name = 'harp' and Initial = 'jm'
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430877(CHEMBL2336480)copy SMILEScopy InChI
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430878(CHEMBL2336474)copy SMILEScopy InChI
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50243007(2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...)copy SMILEScopy InChI
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596239(CHEMBL5189893)copy SMILES
Affinity DataKi:  43nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430876(CHEMBL2336473)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430887(CHEMBL2336479)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430886(CHEMBL2336476)copy SMILEScopy InChI
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430885(CHEMBL2336482)copy SMILEScopy InChI
Affinity DataKi:  94nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430884(CHEMBL2336483)copy SMILEScopy InChI
Affinity DataKi:  157nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430883(CHEMBL2336484)copy SMILEScopy InChI
Affinity DataKi:  201nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430882(CHEMBL2336478)copy SMILEScopy InChI
Affinity DataKi:  252nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430881(CHEMBL2336477)copy SMILEScopy InChI
Affinity DataKi:  277nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430879(CHEMBL2336475)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute of Imaging Science (VUIIS)

Curated by ChEMBL
LigandPNGBDBM50430880(CHEMBL2336481)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z3211ZPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50283472(CHEMBL4160748)copy SMILEScopy InChI
Affinity DataKi:  650nMAssay Description:Displacement of [3H] substance P from recombinant human NK1 receptor expressed in CHO cells after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BN1PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596231(CHEMBL5182783)copy SMILES
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596231(CHEMBL5182783)copy SMILES
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596229(CHEMBL5205163)copy SMILES
Affinity DataIC50: 12nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596229(CHEMBL5205163)copy SMILES
Affinity DataIC50: 12nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596242(CHEMBL5185664)copy SMILES
Affinity DataIC50: 18nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596230(CHEMBL5178468)copy SMILES
Affinity DataIC50: 28nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596230(CHEMBL5178468)copy SMILES
Affinity DataIC50: 28nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596237(CHEMBL5172967)copy SMILES
Affinity DataIC50: 33nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596237(CHEMBL5172967)copy SMILES
Affinity DataIC50: 33nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596237(CHEMBL5172967)copy SMILES
Affinity DataIC50: 42nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596237(CHEMBL5172967)copy SMILES
Affinity DataIC50: 42nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596236(CHEMBL5173887)copy SMILES
Affinity DataIC50: 51nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596236(CHEMBL5173887)copy SMILES
Affinity DataIC50: 52nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596234(CHEMBL5203077)copy SMILES
Affinity DataIC50: 54nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596234(CHEMBL5203077)copy SMILES
Affinity DataIC50: 54nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596239(CHEMBL5189893)copy SMILES
Affinity DataIC50: 71nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596239(CHEMBL5189893)copy SMILES
Affinity DataIC50: 71nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596233(CHEMBL5207446)copy SMILES
Affinity DataIC50: 72nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596233(CHEMBL5207446)copy SMILES
Affinity DataIC50: 72nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
LigandPNGBDBM50596229(CHEMBL5205163)copy SMILES
Affinity DataIC50: 81nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
LigandPNGBDBM50596229(CHEMBL5205163)copy SMILES
Affinity DataIC50: 81nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596232(CHEMBL5185022)copy SMILES
Affinity DataIC50: 120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596232(CHEMBL5185022)copy SMILES
Affinity DataIC50: 123nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596238(CHEMBL5198423)copy SMILES
Affinity DataIC50: 126nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596238(CHEMBL5198423)copy SMILES
Affinity DataIC50: 130nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
LigandPNGBDBM50596242(CHEMBL5185664)copy SMILES
Affinity DataIC50: 228nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596235(CHEMBL5204478)copy SMILES
Affinity DataIC50: 275nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50596235(CHEMBL5204478)copy SMILES
Affinity DataIC50: 280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50283479(CHEMBL4165248)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate preincubated for 15 mins followed by NADPH addition measured after 8 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BN1PubMed
LigandPNGBDBM50596230(CHEMBL5178468)copy SMILES
Affinity DataIC50: 525nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
LigandPNGBDBM50596230(CHEMBL5178468)copy SMILES
Affinity DataIC50: 530nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50596237(CHEMBL5172967)copy SMILES
Affinity DataIC50: 550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F193SZPubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50280374(CHEMBL4174742)copy SMILEScopy InChI
Affinity DataIC50: 650nMAssay Description:Negative allosteric modulation of rat mGlu7 receptor expressed in HEK cells co-expressing Galphai5 assessed as decrease in glutamate-induced thallium...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BN1PubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50283483(CHEMBL2361777)copy SMILEScopy InChI
Affinity DataIC50: 690nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate preincubated for 15 mins followed by NADPH addition measured after 8 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BN1PubMed
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