Affinity DataIC50: 10nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derivedMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derivedMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derivedMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derivedMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against endothelin converting enzyme 1 using bradykinin-derived substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition assay using ECE.More data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human liver microsomes CYP3A4 using testosterone as substrateMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human liver microsomes CYP3A4 using midazolam as substrate preincubated with compound followed by substrate additionMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human liver microsomes CYP3A4 using midazolam as substrateMore data for this Ligand-Target Pair
TargetCytochrome P450 2C19(Homo sapiens (Human))
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human liver microsomes CYP2C19 using S-mephenytoin as substrateMore data for this Ligand-Target Pair
TargetCytochrome P450 2C9(Homo sapiens (Human))
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human liver microsomes CYP2C9 using diclofenac as substrateMore data for this Ligand-Target Pair
TargetCytochrome P450 2B6(Homo sapiens (Human))
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human liver microsomes CYP2B6 using bupropion as substrateMore data for this Ligand-Target Pair
TargetCytochrome P450 2A6(Homo sapiens (Human))
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human liver microsomes CYP2A6 using coumarin as substrateMore data for this Ligand-Target Pair
TargetCytochrome P450 1A2(Homo sapiens (Human))
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Drug Discovery, Bayer AG , Aprather Weg 18a, 42113 Wuppertal, Germany.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human liver microsomes CYP1A2 using phenacetin as substrateMore data for this Ligand-Target Pair
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