Compile Data Set for Download or QSAR
Found 135 with Last Name = 'sun' and Initial = 'jp'
LigandPNGBDBM50250606(CHEMBL4077342)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of STEP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564155(CHEMBL4792956)copy SMILES
Affinity DataKi:  2.20E+3nMAssay Description:Competitive inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) assessed as inhibition of p-nitrophen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564156(CHEMBL4780469)copy SMILES
Affinity DataKi:  2.30E+3nMAssay Description:Competitive inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) assessed as inhibition of p-nitrophen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031906(CHEMBL3360905)copy SMILEScopy InChI
Affinity DataKi:  2.87E+3nMAssay Description:Competitive inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50564157(CHEMBL4792963)copy SMILES
Affinity DataKi:  3.70E+3nMAssay Description:Competitive inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) assessed as inhibition of p-nitrophen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564158(CHEMBL4794022)copy SMILES
Affinity DataKi:  5.40E+3nMAssay Description:Competitive inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) assessed as inhibition of p-nitrophen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50343530(5,7-dichloro-4-((3-(4-methoxyphenylthio)benzyl)(me...)copy SMILEScopy InChI
Affinity DataKi:  5.53E+3nMAssay Description:Competitive inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50441296(CHEMBL2431665 | CHEMBL2431667)copy SMILEScopy InChI
Affinity DataKi:  7.80E+3nMAssay Description:Inhibition of STEP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031908(CHEMBL3360906)copy SMILEScopy InChI
Affinity DataKi:  9.97E+3nMAssay Description:Competitive inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031910(CHEMBL3360908)copy SMILEScopy InChI
Affinity DataKi:  1.03E+4nMAssay Description:Competitive inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031905(CHEMBL3360904)copy SMILEScopy InChI
Affinity DataKi:  1.49E+4nMAssay Description:Competitive inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031907(CHEMBL2337245)copy SMILEScopy InChI
Affinity DataKi:  1.79E+4nMAssay Description:Competitive inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031909(CHEMBL3360907)copy SMILEScopy InChI
Affinity DataKi:  1.92E+4nMAssay Description:Competitive inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50534982(CHEMBL4439458)copy SMILEScopy InChI
Affinity DataKi:  2.16E+4nMAssay Description:Time-dependent irreversible inhibition of N-terminal His-tagged STEP catalytic domain (unknown origin) expressed in Escherichia coli BL21 (DE3) cells...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B0603PubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031904(CHEMBL3360903)copy SMILEScopy InChI
Affinity DataKi:  2.62E+4nMAssay Description:Competitive inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031911(CHEMBL1299903)copy SMILEScopy InChI
Affinity DataKi:  4.10E+4nMAssay Description:Covalent irreversible inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50067512(CHEMBL3401893)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of STEP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031906(CHEMBL3360905)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PTP1B (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50335895(6-hydroxy-3-(1-(4-(naphthalen-1-ylamino)-4-oxobuty...)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of lymphoid-specific tyrosine phosphataseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4QJDPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031906(CHEMBL3360905)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) assessed as re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031916(CHEMBL3360912)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) assessed as re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50564155(CHEMBL4792956)copy SMILES
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031906(CHEMBL3360905)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of VHR (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50564156(CHEMBL4780469)copy SMILES
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50534982(CHEMBL4439458)copy SMILEScopy InChI
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of N-terminal His-tagged STEP catalytic domain (unknown origin) expressed in Escherichia coli BL21 (DE3) cells using p-nitrophenyl phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B0603PubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50564157(CHEMBL4792963)copy SMILES
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of VHR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564158(CHEMBL4794022)copy SMILES
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564164(CHEMBL4794142)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50564157(CHEMBL4792963)copy SMILES
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of LYP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 9(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031906(CHEMBL3360905)copy SMILEScopy InChI
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of MEG2 (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50564157(CHEMBL4792963)copy SMILES
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50335895(6-hydroxy-3-(1-(4-(naphthalen-1-ylamino)-4-oxobuty...)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4QJDPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50564155(CHEMBL4792956)copy SMILES
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50564158(CHEMBL4794022)copy SMILES
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50564156(CHEMBL4780469)copy SMILES
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of LYP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50564157(CHEMBL4792963)copy SMILES
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50534983(CHEMBL4470722)copy SMILEScopy InChI
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of N-terminal His-tagged STEP catalytic domain (unknown origin) expressed in Escherichia coli BL21 (DE3) cells using p-nitrophenyl phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B0603PubMed
LigandPNGBDBM50031906(CHEMBL3360905)copy SMILEScopy InChI
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of STEP (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50564158(CHEMBL4794022)copy SMILES
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of GLEEP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564163(CHEMBL4779840)copy SMILES
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031908(CHEMBL3360906)copy SMILEScopy InChI
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of N-terminal His-tagged Lyp (unknown origin) catalytic domain (1 to 294 residues) expressed in Escherichia coli BL21 (DE3) assessed as re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50564161(CHEMBL4790102)copy SMILES
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 22(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50564155(CHEMBL4792956)copy SMILES
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of LYP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564165(CHEMBL4783271)copy SMILES
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564156(CHEMBL4780469)copy SMILES
Affinity DataIC50: 2.01E+4nMAssay Description:Inhibition of HEPTP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetProtein phosphatase 1A(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50343530(5,7-dichloro-4-((3-(4-methoxyphenylthio)benzyl)(me...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of PPM1A (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
LigandPNGBDBM50564173(CHEMBL4787643)copy SMILES
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
LigandPNGBDBM50564172(CHEMBL4778575)copy SMILES
Affinity DataIC50: 2.46E+4nMAssay Description:Inhibition of N-terminal His-tagged striatal-enriched protein tyrosine phosphatase (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50564156(CHEMBL4780469)copy SMILES
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of VHR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21KHPubMed
TargetTyrosine-protein phosphatase non-receptor type 18(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50031906(CHEMBL3360905)copy SMILEScopy InChI
Affinity DataIC50: 2.64E+4nMAssay Description:Inhibition of PTPN18 (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6TVJPubMed
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