Affinity DataKi: 3.80E+3nMAssay Description:Compound was evaluated to inactivate the bacterial AdoMet-DC; value ranges from 3.8 to 39.6 uMMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Compound was evaluated to inactivate the human AdoMet-DCMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+4nMAssay Description:Compound was evaluated to inactivate the human AdoMet-DC; value ranges from 10.7 to 62.7 uMMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+4nMAssay Description:Compound was evaluated to inactivate the bacterial AdoMet-DC; value ranges from 3.8 to 39.6 uMMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Tested for irreversible inhibitory activity against AdoMet-DC (S-adenosyl-methionine decarboxylase-) isolated from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 3.11E+4nMAssay Description:Compound was evaluated to inactivate the bacterial AdoMet-DCMore data for this Ligand-Target Pair
Affinity DataKi: 2.47E+5nMAssay Description:Compound was evaluated to inactivate the human AdoMet-DCMore data for this Ligand-Target Pair
Affinity DataKi: 4.15E+5nMAssay Description:Tested for irreversible inhibitory activity against AdoMet-DC (S-adenosyl-methionine decarboxylase-) isolated from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 4.78E+5nMAssay Description:Tested for irreversible inhibitory activity against AdoMet-DC (S-adenosyl-methionine decarboxylase-) isolated from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 6.69E+5nMAssay Description:Tested for irreversible inhibitory activity against AdoMet-DC (S-adenosyl-methionine decarboxylase-) isolated from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 9.60E+5nMAssay Description:Tested for irreversible inhibitory activity against AdoMet-DC (S-adenosyl-methionine decarboxylase-) isolated from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+6nMAssay Description:Tested for irreversible inhibitory activity against AdoMet-DC (S-adenosyl-methionine decarboxylase-) isolated from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+6nMAssay Description:Tested for irreversible inhibitory activity against AdoMet-DC (S-adenosyl-methionine decarboxylase-) isolated from Escherichia coliMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 1.64E+3nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 3.28E+3nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Compound was evaluated for its inhibitory activity against AdoMet-DC from Escherichia coliMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 9.95E+3nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 1.47E+4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 1.76E+4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Compound was evaluated to inactivate the bacterial AdoMet-DCMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Cambridge NeuroScience Inc.
Curated by ChEMBL
Cambridge NeuroScience Inc.
Curated by ChEMBL
Affinity DataIC50: 5.30E+4nMAssay Description:In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1)More data for this Ligand-Target Pair
Affinity DataIC50: 1.79E+5nMAssay Description:Compound was evaluated for its inhibitory activity against AdoMet-DC from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 2.05E+5nMAssay Description:Compound was evaluated for its inhibitory activity against AdoMet-DC from Escherichia coliMore data for this Ligand-Target Pair