BindingDB PrimarySearch_ki

Found 478 with Last Name = 'li' and Initial = 'jq'

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207116(CHEMBL3905247 | US9550741, I-4)copy SMILEScopy InChI

Ki: 0.0290nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207143(CHEMBL3966842 | US9550741, II-1)copy SMILEScopy InChI

Ki: 0.0430nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207162(CHEMBL3918755 | US9550741, IV-1)copy SMILEScopy InChI

Ki: 0.0430nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207155(CHEMBL3895540)copy SMILEScopy InChI

Ki: 0.0460nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207141(CHEMBL3920252)copy SMILEScopy InChI

Ki: 0.0470nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207148(CHEMBL3932186)copy SMILEScopy InChI

Ki: 0.0510nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207154(CHEMBL3902496)copy SMILEScopy InChI

Ki: 0.0520nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207113(CHEMBL3896937 | US9550741, IV-3)copy SMILEScopy InChI

Ki: 0.0550nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207094(CHEMBL3976282 | US9550741, I-2)copy SMILEScopy InChI

Ki: 0.0560nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207150(CHEMBL3933256)copy SMILEScopy InChI

Ki: 0.0580nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207158(CHEMBL3982486 | US9550741, III-2)copy SMILEScopy InChI

Ki: 0.0580nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207115(CHEMBL3948056)copy SMILEScopy InChI

Ki: 0.0620nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 1A(Homo sapiens (Human))TBA

PNG

BDBM50607169(CHEMBL5220371)copy SMILES

Ki: 0.0690nMMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2ZC8701PubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50443101(Cariprazine | RGH-188)copy SMILEScopy InChI

Ki: 0.0850nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2BZ69PBPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207112(CHEMBL3967779)copy SMILEScopy InChI

Ki: 0.0900nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207114(CHEMBL3892440)copy SMILEScopy InChI

Ki: 0.0950nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50443101(Cariprazine | RGH-188)copy SMILEScopy InChI

Ki: 0.0960nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 1A(Homo sapiens (Human))TBA

PNG

BDBM50607170(CHEMBL5220872)copy SMILES

Ki: 0.0970nMMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2ZC8701PubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207145(CHEMBL3946995 | US9550741, I-1)copy SMILEScopy InChI

Ki: 0.130nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207160(CHEMBL3962525)copy SMILEScopy InChI

Ki: 0.140nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207113(CHEMBL3896937 | US9550741, IV-3)copy SMILEScopy InChI

Ki: 0.140nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

Alpha-1A adrenergic receptor(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL

PNG

BDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)copy SMILEScopy InChI

Ki: 0.150nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor (unknown origin) in cerebral cortex membranes after 60 mins by TopCount scintillation counting ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed DrugBank

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207094(CHEMBL3976282 | US9550741, I-2)copy SMILEScopy InChI

Ki: 0.150nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207142(CHEMBL3973487)copy SMILEScopy InChI

Ki: 0.160nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207144(CHEMBL3940712 | US9550741, IV-11)copy SMILEScopy InChI

Ki: 0.180nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207110(CHEMBL3923240 | US9550741, III-15)copy SMILEScopy InChI

Ki: 0.180nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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CHEMBL PC cid PC sid Patents Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207146(CHEMBL3929168)copy SMILEScopy InChI

Ki: 0.190nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(2) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207094(CHEMBL3976282 | US9550741, I-2)copy SMILEScopy InChI

Ki: 0.190nMAssay Description:Displacement of [3H]spiperone from recombinant human D2L receptor expressed in CHO cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207161(CHEMBL3950977 | US9550741, I-19)copy SMILEScopy InChI

Ki: 0.190nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

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CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 1A(Homo sapiens (Human))TBA

PNG

BDBM50529312(CHEMBL4444213)copy SMILEScopy InChI

Ki: 0.200nMMore data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2ZC8701PubMed

5-hydroxytryptamine receptor 1A(Homo sapiens (Human))TBA

PNG

BDBM50207158(CHEMBL3982486 | US9550741, III-2)copy SMILEScopy InChI

Ki: 0.200nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 1A(Homo sapiens (Human))TBA

PNG

BDBM50151982(5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1...)copy SMILEScopy InChI

Ki: 0.200nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin) expressed in HEK293 cells membranes incubated for 60 mins by scintillation counti...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2DR2ZZTPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207092(CHEMBL3891773)copy SMILEScopy InChI

Ki: 0.210nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

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CHEMBL PC cid PC sid Patents Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(2) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207156(CHEMBL3938210 | US9550741, I-3)copy SMILEScopy InChI

Ki: 0.210nMAssay Description:Displacement of [3H]spiperone from recombinant human D2L receptor expressed in CHO cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207147(CHEMBL3956720)copy SMILEScopy InChI

Ki: 0.210nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207162(CHEMBL3918755 | US9550741, IV-1)copy SMILEScopy InChI

Ki: 0.210nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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CHEMBL PC cid PC sid

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207108(CHEMBL3920432)copy SMILEScopy InChI

Ki: 0.220nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207145(CHEMBL3946995 | US9550741, I-1)copy SMILEScopy InChI

Ki: 0.230nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

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CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207141(CHEMBL3920252)copy SMILEScopy InChI

Ki: 0.240nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207117(CHEMBL3970746)copy SMILEScopy InChI

Ki: 0.240nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207157(CHEMBL3903560)copy SMILEScopy InChI

Ki: 0.240nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207115(CHEMBL3948056)copy SMILEScopy InChI

Ki: 0.260nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL

PNG

BDBM50464861(CHEMBL4291322)copy SMILEScopy InChI

Ki: 0.260nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Details Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207090(CHEMBL3913691)copy SMILEScopy InChI

Ki: 0.270nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

PDB
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Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207114(CHEMBL3892440)copy SMILEScopy InChI

Ki: 0.280nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207156(CHEMBL3938210 | US9550741, I-3)copy SMILEScopy InChI

Ki: 0.290nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207112(CHEMBL3967779)copy SMILEScopy InChI

Ki: 0.290nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207143(CHEMBL3966842 | US9550741, II-1)copy SMILEScopy InChI

Ki: 0.300nMAssay Description:Displacement of [3H]ketanserin from recombinant human 5-HT2A receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting meth...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(2) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207155(CHEMBL3895540)copy SMILEScopy InChI

Ki: 0.300nMAssay Description:Displacement of [3H]spiperone from recombinant human D2L receptor expressed in CHO cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

D(3) dopamine receptor(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL

PNG

BDBM50207157(CHEMBL3903560)copy SMILEScopy InChI

Ki: 0.310nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2GH9KXPPubMed

Displayed 1 to 50 (of 478 total ) | Next | Last >>

Targets 17 ▿
- 5-hydroxytryptamine receptor 1A 94
- Sodium-dependent serotonin transporter 74
- D(2) dopamine receptor 62
- D(3) dopamine receptor 61
- 5-hydroxytryptamine receptor 2A 46
- 5-hydroxytryptamine receptor 7 27
- Rho-associated protein kinase 2 25
- Sodium-dependent noradrenaline transporter 24
- Sodium-dependent dopamine transporter 18
- Histamine H1 receptor 11
- Mitogen-activated protein kinase kinase kinase 5 10
- Protein kinase C alpha type 10
- Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor 8
- Potassium voltage-gated channel subfamily H member 2 4
- Alpha-1A adrenergic receptor 2
- D(1A) dopamine receptor 1
- Metallo-beta-lactamase type 2 1
- ...
Publications 10 ▿
- Eur J Med Chem 123: 332-353 (2016) 169
- Eur J Med Chem 144: 701-715 (2018) 46
- Eur J Med Chem 86: 219-34 (2014) 41
- Bioorg Med Chem Lett 29: (2019) 33
- J Nat Prod 81: 949-956 (2018) 30
- Eur J Med Chem 54: 123-36 (2012) 25
- Bioorg Med Chem Lett 27: 5420-5423 (2017) 21
- J Nat Prod 81: 394-399 (2018) 10
- Bioorg Med Chem Lett 29: (2019) 9
- J Nat Prod 81: 2120-2124 (2018) 5
Institutions 5 ▿
- [Shanghai Jiao Tong University] 169
- [Shanghai Institute of Pharmaceutical Industry] 133
- [Zhejiang University] 45
- [China State Institute of Pharmaceutical Industry] 33
- [China Pharmaceutical University] 9
Affinity: 0.029 to 1.0E+5 nM▿
- Ki 297
- IC50 171
- EC50 10
- Affinity ≤ nM
Xtal structures: 6
Docked structures: 0
Catalog Cmpds: 18