Compile Data Set for Download or QSAR
Found 120 with Last Name = 'trojanowski' and Initial = 'jq'
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50101410((trans,trans)-1-bromo-2,5-bis-(3-hydroxycarbonyl-4...)copy SMILEScopy InChI
Affinity DataKi:  0.110nMAssay Description:Inhibitory activity against binding of [125I]-IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22J6B4ZPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50101411(5-[2-bromo-4-(3-carboxy-4-hydroxyphenethyl)pheneth...)copy SMILEScopy InChI
Affinity DataKi:  0.130nMAssay Description:Inhibitory activity against binding of [125I]-IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22J6B4ZPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100131(5-(Biphenyl-4-ylazo)-bis (2-hydroxy-benzoic acid)(...)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Inhibitory activity against binding of [125I]-IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22J6B4ZPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100131(5-(Biphenyl-4-ylazo)-bis (2-hydroxy-benzoic acid)(...)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100135((E,E)-1-iodo-2,5-bis-(3-hydroxycarbonyl-4-methoxy)...)copy SMILEScopy InChI
Affinity DataKi:  0.170nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100135((E,E)-1-iodo-2,5-bis-(3-hydroxycarbonyl-4-methoxy)...)copy SMILEScopy InChI
Affinity DataKi:  0.170nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50101413(5-[2-bromo-4-(3-carboxy-4-hydroxyphenethyl)pheneth...)copy SMILEScopy InChI
Affinity DataKi:  0.190nMAssay Description:Inhibitory activity against binding of [125I]-IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22J6B4ZPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50101412(5-[2-bromo-4-(3-carboxy-4-hydroxyphenethyl)pheneth...)copy SMILEScopy InChI
Affinity DataKi:  0.270nMAssay Description:Inhibitory activity against binding of [125I]-IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22J6B4ZPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100131(5-(Biphenyl-4-ylazo)-bis (2-hydroxy-benzoic acid)(...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Inhibition constant of compound on ligand binding to aggregates of Amyloid beta was measured by comparing with [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100130(4-(6-Iodobenzo[d]thiazol-2-yl)-N,N-dimethylaniline...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100130(4-(6-Iodobenzo[d]thiazol-2-yl)-N,N-dimethylaniline...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100132(6-Bromo-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-ben...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100132(6-Bromo-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-ben...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100133(CHEMBL55401 | [4-(6-Bromo-benzothiazol-2-yl)-pheny...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100133(CHEMBL55401 | [4-(6-Bromo-benzothiazol-2-yl)-pheny...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100136(6-Iodo-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-benz...)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100136(6-Iodo-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-benz...)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100134(2-(4-Dimethylamino-phenyl)-3,6-dimethyl-benzothiaz...)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100134(2-(4-Dimethylamino-phenyl)-3,6-dimethyl-benzothiaz...)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100135((E,E)-1-iodo-2,5-bis-(3-hydroxycarbonyl-4-methoxy)...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100131(5-(Biphenyl-4-ylazo)-bis (2-hydroxy-benzoic acid)(...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition constant for amyloid beta compared to [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM26193(2-Hydroxybenzoate, I | 2-hydroxybenzoic acid | CHE...)copy SMILEScopy InChI
Affinity DataKi: >1.80E+3nMAssay Description:Inhibitory activity against binding of [125I]-IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22J6B4ZPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100130(4-(6-Iodobenzo[d]thiazol-2-yl)-N,N-dimethylaniline...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100133(CHEMBL55401 | [4-(6-Bromo-benzothiazol-2-yl)-pheny...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100133(CHEMBL55401 | [4-(6-Bromo-benzothiazol-2-yl)-pheny...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100130(4-(6-Iodobenzo[d]thiazol-2-yl)-N,N-dimethylaniline...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100131(5-(Biphenyl-4-ylazo)-bis (2-hydroxy-benzoic acid)(...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition constant of compound on ligand binding to aggregates of Amyloid beta was measured by comparing with [125I]-TZDMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100132(6-Bromo-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-ben...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100132(6-Bromo-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-ben...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100136(6-Iodo-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-benz...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100134(2-(4-Dimethylamino-phenyl)-3,6-dimethyl-benzothiaz...)copy SMILEScopy InChI
Affinity DataKi: >9.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50100134(2-(4-Dimethylamino-phenyl)-3,6-dimethyl-benzothiaz...)copy SMILEScopy InChI
Affinity DataKi: >9.00E+3nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HV8PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50026750(CHEMBL3354618)copy SMILEScopy InChI
Affinity DataIC50: 0.0150nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09HFPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50026748(CHEMBL3354616)copy SMILEScopy InChI
Affinity DataIC50: 0.0520nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09HFPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50058027(CHEMBL29374)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human TP receptor expressed in QBI-HEK 293A cells assessed as IP3 metabolite level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8VJ5PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353639(CHEMBL1829806)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50026760(CHEMBL3354614)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09HFPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353632(CHEMBL1829812)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50026761(CHEMBL3354615)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09HFPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353635(CHEMBL1829801)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353643(CHEMBL1829808)copy SMILEScopy InChI
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50026758(CHEMBL3335473)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09HFPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50026759(CHEMBL3354613)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09HFPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50026753(S-18886 | Terutroban)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09HFPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353645(CHEMBL1829810)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353640(CHEMBL65121)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50026751(CHEMBL3354619)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09HFPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353632(CHEMBL1829812)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Antagonist activity at human prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353638(CHEMBL1829805)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50058026(CHEMBL3326602)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of human TP receptor expressed in QBI-HEK 293A cells assessed as IP3 metabolite level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8VJ5PubMed
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