Compile Data Set for Download or QSAR
Found 523 with Last Name = 'medina' and Initial = 'jr'
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383996(CHEMBL2032134)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383999(CHEMBL2032137)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383966(CHEMBL2032148)copy SMILEScopy InChI
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383998(CHEMBL2032136)copy SMILEScopy InChI
Affinity DataIC50: 0.190nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50384000(CHEMBL2032138)copy SMILEScopy InChI
Affinity DataIC50: 0.190nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383997(CHEMBL2032135)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396532(CHEMBL2171126)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396540(CHEMBL2171143)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396542(CHEMBL2171141)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396539(CHEMBL2171144)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396536(CHEMBL2171122)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383994(CHEMBL2032132)copy SMILEScopy InChI
Affinity DataIC50: 0.220nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383987(CHEMBL2032125)copy SMILEScopy InChI
Affinity DataIC50: 0.260nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383982(CHEMBL2032119)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383988(CHEMBL2032126)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383995(CHEMBL2032133)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396533(CHEMBL2171125)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383993(CHEMBL2032131)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383968(CHEMBL2032140)copy SMILEScopy InChI
Affinity DataIC50: 0.350nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50384003(CHEMBL2032142)copy SMILEScopy InChI
Affinity DataIC50: 0.350nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50384002(CHEMBL2032141)copy SMILEScopy InChI
Affinity DataIC50: 0.370nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383972(CHEMBL2032146)copy SMILEScopy InChI
Affinity DataIC50: 0.380nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396544(CHEMBL2171139)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396534(CHEMBL2171124)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396534(CHEMBL2171124)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of GST-tagged PERK cytoplasmic domain (536 to 1116) (unknown origin) assessed as biotinylated His6-tagged EIF2alpha phosphorylation preinc...More data for this Ligand-Target Pair
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383969(CHEMBL2032143)copy SMILEScopy InChI
Affinity DataIC50: 0.410nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383980(CHEMBL2032117)copy SMILEScopy InChI
Affinity DataIC50: 0.430nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383992(CHEMBL2032130)copy SMILEScopy InChI
Affinity DataIC50: 0.440nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383965(CHEMBL2032129)copy SMILEScopy InChI
Affinity DataIC50: 0.460nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383967(CHEMBL2032122)copy SMILEScopy InChI
Affinity DataIC50: 0.480nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396535(CHEMBL2171123)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50442165(CHEMBL2441341)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged PERK cytoplasmic domain (536 to 1116) (unknown origin) assessed as biotinylated His6-tagged EIF2alpha phosphorylation preinc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X597XPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383981(CHEMBL2032118)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50442162(CHEMBL2441342)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged PERK cytoplasmic domain (536 to 1116) (unknown origin) assessed as biotinylated His6-tagged EIF2alpha phosphorylation preinc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X597XPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383986(CHEMBL2032124)copy SMILEScopy InChI
Affinity DataIC50: 0.510nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383985(CHEMBL2032123)copy SMILEScopy InChI
Affinity DataIC50: 0.520nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Staphylococcus aureus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383996(CHEMBL2032134)copy SMILEScopy InChI
Affinity DataIC50: 0.520nMAssay Description:Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383984(CHEMBL2032121)copy SMILEScopy InChI
Affinity DataIC50: 0.540nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396548(CHEMBL2171135)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50341250(CHEMBL1765751 | N-{(3R,5R)-1-[2-Amino-6-(3-amino-1...)copy SMILEScopy InChI
Affinity DataIC50: 0.631nMAssay Description:Inhibition of PDK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ406QPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383989(CHEMBL2032127)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396543(CHEMBL2171140)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383978(CHEMBL2032115)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383973(CHEMBL2032147)copy SMILEScopy InChI
Affinity DataIC50: 0.720nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383971(CHEMBL2032145)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50341249(1,1-Dimethylethyl{(3R,5R)-1-[2-Amino-6-(3-amino-1H...)copy SMILEScopy InChI
Affinity DataIC50: 0.794nMAssay Description:Inhibition of PDK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ406QPubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383976(CHEMBL2032113)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50442166(CHEMBL2441340)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Inhibition of GST-tagged PERK cytoplasmic domain (536 to 1116) (unknown origin) assessed as biotinylated His6-tagged EIF2alpha phosphorylation preinc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X597XPubMed
TargetPeptide deformylase(Staphylococcus aureus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50383999(CHEMBL2032137)copy SMILEScopy InChI
Affinity DataIC50: 0.860nMAssay Description:Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64K3VPubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50396537(CHEMBL2171121 | D3RKN_50)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of GST tagged PERK cytoplasmic domain mediated EIF2alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222VWPPubMed
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