Affinity DataIC50: 20nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Calpain 1 by [3H]-acetyl-casein assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:In vitro inhibitory activity against cathepsin LMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro inhibitory activity against Cathepsin BMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibitory activity against human erythrocyte Calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+4nMAssay Description:In vitro inhibitory activity against Cathepsin BMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:In vitro inhibitory activity against cathepsin LMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 314nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 6.30nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 292nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 176nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 268nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 145nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 291nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 590nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 82nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Genzyme Corp.
Curated by ChEMBL
Genzyme Corp.
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Effective concentration for cellular chloride transport in C127 mouse epithelial cell transfected with recombinant Delta F508 CFTRMore data for this Ligand-Target Pair