Affinity DataKi: 6.30nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 1.59E+3nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 3.16E+3nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: <2.51E+4nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: <2.51E+4nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium concentrati...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
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