Compile Data Set for Download or QSAR
Found 135 with Last Name = 'brozinick' and Initial = 'jt'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157059((S)-3-{4-[3-(4-Benzoyl-phenoxy)-propoxy]-phenyl}-2...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157055((S)-3-{4-[3-(4-Benzoyl-phenoxy)-propoxy]-3-chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetSerine palmitoyltransferase 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50535848(CHEMBL4584997)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human SPT1 expressed in microsomes of HEK293 cells incubated for 1hr by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4FR1PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157057((S)-2-Methoxy-3-{4-[5-(4-phenoxy-phenoxy)-pent-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195706(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-(p...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TNKPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157058((S)-2-Methoxy-3-{3-methoxy-4-[3-(4-phenoxy-phenoxy...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157060((S)-2-Methoxy-3-{4-[4-(4-phenoxy-phenoxy)-but-1-yn...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195704(3-(2-(isobutoxycarbonyl)-5-(2-(5-methyl-2-phenylox...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TNKPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157061((S)-3-{4-[3-(Biphenyl-4-yloxy)-propoxy]-phenyl}-2-...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TNKPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195708(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195703(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TNKPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50085044((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195716(3-{4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195714(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195705(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TNKPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157056((S)-2-Methoxy-3-{4-[3-(4-phenoxy-phenoxy)-propoxy]...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157054((S)-2-Ethoxy-3-{4-[3-(4-phenoxy-phenoxy)-propoxy]-...)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TNKPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195715(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195713(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetSerine palmitoyltransferase 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50535847(CHEMBL4541898)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of human SPT1 expressed in microsomes of HEK293 cells incubated for 1hr by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4FR1PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 67nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195707(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195710(3-(2-((benzyloxycarbonyl)methyl)-4-(2-(5-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50195714(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 146nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195712(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)copy SMILEScopy InChI
Affinity DataIC50: 161nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50157055((S)-3-{4-[3-(4-Benzoyl-phenoxy)-propoxy]-3-chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 309nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50195710(3-(2-((benzyloxycarbonyl)methyl)-4-(2-(5-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 441nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50195716(3-{4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)copy SMILEScopy InChI
Affinity DataIC50: 449nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50157059((S)-3-{4-[3-(4-Benzoyl-phenoxy)-propoxy]-phenyl}-2...)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50195715(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 516nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50157061((S)-3-{4-[3-(Biphenyl-4-yloxy)-propoxy]-phenyl}-2-...)copy SMILEScopy InChI
Affinity DataIC50: 568nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195709(3-(2-((3-benzylureido)methyl)-4-(2-(5-methyl-2-phe...)copy SMILEScopy InChI
Affinity DataIC50: 706nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50157057((S)-2-Methoxy-3-{4-[5-(4-phenoxy-phenoxy)-pent-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 770nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50157060((S)-2-Methoxy-3-{4-[4-(4-phenoxy-phenoxy)-but-1-yn...)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+3nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50085044((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.22E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TNKPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.29E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TNKPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50157058((S)-2-Methoxy-3-{3-methoxy-4-[3-(4-phenoxy-phenoxy...)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157061((S)-3-{4-[3-(Biphenyl-4-yloxy)-propoxy]-phenyl}-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.39E+3nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor deltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50195708(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0FSCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157055((S)-3-{4-[3-(4-Benzoyl-phenoxy)-propoxy]-3-chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.51E+3nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor deltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157054((S)-2-Ethoxy-3-{4-[3-(4-phenoxy-phenoxy)-propoxy]-...)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+3nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor deltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly and Co

Curated by ChEMBL
LigandPNGBDBM50157054((S)-2-Ethoxy-3-{4-[3-(4-phenoxy-phenoxy)-propoxy]-...)copy SMILEScopy InChI
Affinity DataIC50: 1.69E+3nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157056((S)-2-Methoxy-3-{4-[3-(4-phenoxy-phenoxy)-propoxy]...)copy SMILEScopy InChI
Affinity DataIC50: 1.92E+3nMAssay Description:Mean inhibitory concentration against human peroxisome proliferator-activated receptor deltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30T6PubMed
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