Affinity DataIC50: 410nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory concentration against wild type HIV-1 reverse transcriptase (RT) using poly rC.dG as the template or primerMore data for this Ligand-Target Pair
Affinity DataIC50: 3.15E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.45E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibitory concentration against wild type HIV-1 reverse transcriptase (RT) using poly rC.dG as the template or primerMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory concentration against wild type HIV-1 reverse transcriptase (RT) using poly rC.dG as the template or primerMore data for this Ligand-Target Pair
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.62E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibitory concentration against wild type HIV-1 reverse transcriptase (RT) using poly rC.dG as the template or primerMore data for this Ligand-Target Pair
Affinity DataIC50: 6.09E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibitory concentration against wild type HIV-1 reverse transcriptase (RT) using poly rC.dG as the template or primerMore data for this Ligand-Target Pair
Affinity DataIC50: 6.34E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibitory concentration against wild type HIV-1 reverse transcriptase (RT) using poly rC.dG as the template or primerMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory concentration against wild type HIV-1 reverse transcriptase (RT) using poly rC.dG as the template or primerMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibitory concentration against wild type HIV-1 reverse transcriptase (RT) using poly rC.dG as the template or primerMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibitory concentration against wild type HIV-1/138Lys reverse transcriptase (RT) using [3H]dGTP as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against wild type HIV-1/138Lys reverse transcriptase (RT) using [3H]dGTP as a radioligandMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against wild type HIV-1/138Lys reverse transcriptase (RT) using [3H]dGTP as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+5nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 2.93E+5nMAssay Description:Inhibitory concentration against wild type HIV-1/138Lys reverse transcriptase (RT) using [3H]dGTP as a radioligandMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 3.12E+5nMAssay Description:Inhibitory concentration against wild type HIV-1/138Lys reverse transcriptase (RT) using [3H]dGTP as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.33E+5nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.33E+5nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.33E+5nMAssay Description:Inhibition of HIV1 recombinant integrase by electrochemiluminescent-based high-throughput strand transfer assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 3.94E+5nMAssay Description:Inhibitory concentration against wild type HIV-1/138Lys reverse transcriptase (RT) using [3H]dGTP as a radioligandMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 4.37E+5nMAssay Description:Inhibitory concentration against wild type HIV-1/138Lys reverse transcriptase (RT) using [3H]dGTP as a radioligandMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Instituto de Química Médica (C.S.I.C.)
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory concentration against wild type HIV-1/138Lys reverse transcriptase (RT) using [3H]dGTP as a radioligandMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataKd: >6.00E+4nMAssay Description:Binding affinity to HIV1 reverse transcriptase M184V mutant assessed as L-3'-azido-NTP incorporation in nascent DNAMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataKd: 2.10E+3nMAssay Description:Binding affinity to HIV1 reverse transcriptase assessed as L-3'-azido-NTP incorporation in nascent DNAMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataKd: 2.50E+3nMAssay Description:Binding affinity to HIV1 reverse transcriptase M184V mutant assessed as L-3'-azido-NTP incorporation in nascent DNAMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataKd: 230nMAssay Description:Binding affinity to HIV1 reverse transcriptase assessed as L-3'-azido-NTP incorporation in nascent DNAMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataKd: 3.00E+3nMAssay Description:Binding affinity to HIV1 reverse transcriptase M184V mutant assessed as L-3'-azido-NTP incorporation in nascent DNAMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Binding affinity to HIV1 reverse transcriptase M184V mutant assessed as L-3'-azido-NTP incorporation in nascent DNAMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)