Affinity DataKi: 300nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Mixed inhibition of equine serum BChE using S-butyrylthiocholine chloride as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 4.33E+3nMAssay Description:Mixed inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 5.20E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 5.40E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 5.50E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 5.70E+3nMAssay Description:Inhibition of Bcl-xL (unknown origin)/Bak interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 ...More data for this Ligand-Target Pair
Affinity DataKi: 5.86E+3nMAssay Description:Mixed inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.72E+3nMAssay Description:Mixed-type inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine chloride as substrate measured after...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 7.20E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 7.30E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 8.20E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 8.30E+3nMAssay Description:Inhibition of Bcl-xL (unknown origin)/Bak interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 ...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 8.50E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 8.60E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 9.00E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 9.20E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 9.60E+3nMAssay Description:Inhibition of Bcl-xL (unknown origin)/Bak interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.08E+4nMAssay Description:Displacement of fluorescent-tagged BH3 domain of Bak from Bcl-xL by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+4nMAssay Description:Mixed inhibition of equine serum BChE using S-butyrylthiocholine chloride as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 1.66E+4nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 1.74E+4nMAssay Description:Inhibition of Bcl-xL (unknown origin)/Bak interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 ...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Universit£ Paris-Saclay
Curated by ChEMBL
Universit£ Paris-Saclay
Curated by ChEMBL
Affinity DataKi: 1.89E+4nMAssay Description:Inhibition of Mcl-1 (unknown origin)/Bid interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Inhibition of Bcl-xL (unknown origin)/Bak interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 ...More data for this Ligand-Target Pair
Affinity DataKi: 2.01E+4nMAssay Description:Inhibition of Bcl-xL (unknown origin)/Bak interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 ...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of Bcl2 (unknown origin)/Bim interaction preincubated for 5 mins followed by fluorescein-labeled peptide addition and measured after 10 mi...More data for this Ligand-Target Pair