Affinity DataIC50: 0.300nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc
Curated by ChEMBL
LifeArc
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc
Curated by ChEMBL
LifeArc
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant C-terminal His10-tagged human Hepsin (R45 to L17 residues) D161E/ R162K double mutant expressed in mouse NS0 cells using Bo...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc
Curated by ChEMBL
LifeArc
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc
Curated by ChEMBL
LifeArc
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
MRC Technology
Curated by ChEMBL
MRC Technology
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc
Curated by ChEMBL
LifeArc
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair