Compile Data Set for Download or QSAR
Found 269 with Last Name = 'birchall' and Initial = 'k'
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467114(CHEMBL4285682)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467117(CHEMBL4288816)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467123(CHEMBL4288103)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467126(CHEMBL4286880)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467122(CHEMBL4279865)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401928(CHEMBL2207195)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401907(CHEMBL2207181)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc

Curated by ChEMBL
LigandPNGBDBM50507968(CHEMBL4444153)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2269PubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467128(CHEMBL4286841)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401915(CHEMBL2207212)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401913(CHEMBL2207214)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401927(CHEMBL2207199)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401903(CHEMBL2207194)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50182362(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc

Curated by ChEMBL
LigandPNGBDBM105071(US8569281, 39)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2269PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401918(CHEMBL2207209)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401914(CHEMBL2207213)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine protease hepsin(Homo sapiens (Human))
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant C-terminal His10-tagged human Hepsin (R45 to L17 residues) D161E/ R162K double mutant expressed in mouse NS0 cells using Bo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3VVTPubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401900(CHEMBL2207198)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401902(CHEMBL2207196)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467127(CHEMBL4284547)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50168171(4-(2-(4-fluorophenyl)-5-(1-methylpiperidin-4-yl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467124(CHEMBL4283774)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401910(CHEMBL2207217)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401911(CHEMBL2207216)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401922(CHEMBL2207204)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401920(CHEMBL2207206)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401917(CHEMBL2207210)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401899(CHEMBL2207208)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401908(CHEMBL2207180)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401906(CHEMBL2207187)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401901(CHEMBL2207197)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613268(CHEMBL5275681)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401924(CHEMBL2207202)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467116(CHEMBL4287934)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401912(CHEMBL2207215)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401909(CHEMBL2207218)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401916(CHEMBL2207211)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc

Curated by ChEMBL
LigandPNGBDBM50507979(CHEMBL4589022)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2269PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401905(CHEMBL2207192)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613266(CHEMBL5268562)copy SMILES
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc

Curated by ChEMBL
LigandPNGBDBM50507672(CHEMBL4460272)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2269PubMed
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401900(CHEMBL2207198)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of MARK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401926(CHEMBL2207200)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613282(CHEMBL5270264)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
LifeArc

Curated by ChEMBL
LigandPNGBDBM50507981(CHEMBL4561299)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD2269PubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467121(CHEMBL4282026)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401925(CHEMBL2207201)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50401921(CHEMBL2207205)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4S45PubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
LifeArc

Curated by ChEMBL
LigandPNGBDBM50467119(CHEMBL4281827)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z473BPubMed
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