Compile Data Set for Download or QSAR
Found 74 with Last Name = 'korpis' and Initial = 'k'
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50125099(1-Benzyl-4-(4-methoxy-benzyl)-piperazine | 1-benzy...)copy SMILEScopy InChI
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XM7PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181060(CHEMBL3817940)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50009304(CHEMBL3233531)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181297(CHEMBL3819489)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181054(CHEMBL3819146)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50009303(CHEMBL3233530)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50009302(CHEMBL3233529)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181054(CHEMBL3819146)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181300(CHEMBL3819437)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181299(CHEMBL3819331)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181301(CHEMBL3819395)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50445477(CHEMBL3104856)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XM7PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50445477(CHEMBL3104856)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50009301(CHEMBL3233528)copy SMILEScopy InChI
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50009305(CHEMBL3233532)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181301(CHEMBL3819395)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50001028((+)-PENTAZOCINE | (-)-pentazocine | (2R,6R,11R)-6,...)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50035131((+)-(6R,11S)-6,11-dimethyl-3-(3-methyl-but-2-enyl)...)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181297(CHEMBL3819489)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181060(CHEMBL3817940)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181055(CHEMBL3819463)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181055(CHEMBL3819463)copy SMILEScopy InChI
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50009305(CHEMBL3233532)copy SMILEScopy InChI
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cell membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181300(CHEMBL3819437)copy SMILEScopy InChI
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181113(CHEMBL3818112)copy SMILEScopy InChI
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181113(CHEMBL3818112)copy SMILEScopy InChI
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50009304(CHEMBL3233531)copy SMILEScopy InChI
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cell membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50445476(CHEMBL3104857)copy SMILEScopy InChI
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain cortex membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50445476(CHEMBL3104857)copy SMILEScopy InChI
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XM7PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181130(CHEMBL3818532)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181059(CHEMBL3819588)copy SMILEScopy InChI
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181057(CHEMBL3819457)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181056(CHEMBL3818546)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50257493((R)-(1-benzyl-4-(4-methoxybenzyl)piperazin-2-yl)me...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Binding affinity to sigma-1 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XM7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50048866(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-na...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Binding affinity to sigma-1 receptor in human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XM7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181130(CHEMBL3818532)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181061(CHEMBL3819557)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50009301(CHEMBL3233528)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cell membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181299(CHEMBL3819331)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50181058(CHEMBL3818045)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50009302(CHEMBL3233529)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cell membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181056(CHEMBL3818546)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50009306(CHEMBL3233533)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cell membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181059(CHEMBL3819588)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50181057(CHEMBL3819457)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Displacement of [3H](+)-Pentazocine from sigma 1 receptor in human RPMI8226 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12KNPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50009303(CHEMBL3233530)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cell membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50445476(CHEMBL3104857)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cell membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T15562PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of M£nster

Curated by ChEMBL
LigandPNGBDBM50445476(CHEMBL3104857)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XM7PubMed
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