Compile Data Set for Download or QSAR
Found 105 with Last Name = 'kunishiro' and Initial = 'k'
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296994(CHEMBL561939 | N-(5-Methanesulfonylamino-4,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50263150(CHEMBL513892 | N-(4,6-dimethyl-1-octylindolin-7-yl...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297009(CHEMBL550526 | N-(1-decyl-4,6-dimethylindolin-7-yl...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297008(CHEMBL558454 | N-(1-heptyl-4,6-dimethylindolin-7-y...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297017(CHEMBL555564 | N-[1-(Cyclobutylmethyl)-5-methanesu...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297014(CHEMBL559117 | N-[5-Methanesulfonylamino-4,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296993(CHEMBL557522 | N-(1-Hexyl-5-methanesulfonylamino-4...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296992(CHEMBL559879 | N-(5-Methanesulfonylamino-4,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297022(CHEMBL564138 | N-(1-Butyl-5-methanesulfonylamino-4...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297010(CHEMBL561477 | N-(1-dodecyl-4,6-dimethylindolin-7-...)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297013(CHEMBL554505 | N-[1-(2,2-Dimethylpropyl)-5-methane...)copy SMILEScopy InChI
Affinity DataIC50: 61nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297007(CHEMBL561074 | N-(1-hexyl-4,6-dimethylindolin-7-yl...)copy SMILEScopy InChI
Affinity DataIC50: 67nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297015(CHEMBL559318 | N-[5-Methanesulfonylamino-4,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296991(CHEMBL551271 | N-(1-Butyl-5-methanesulfonylamino-4...)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297012(CHEMBL549649 | N-[5-Methanesulfonylamino-4,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297018(CHEMBL556503 | N-[1-(Cyclopentyl)-5-methanesulfony...)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297006(CHEMBL563443 | N-(4,6-dimethyl-1-pentylindolin-7-y...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297025(CHEMBL561135 | N-(5,7-dimethyl-6-(methylsulfonamid...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297016(CHEMBL560997 | N-[1-(Cyclopropylmethyl)-5-methanes...)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297005(CHEMBL538381 | N-(1-butyl-4,6-dimethylindolin-7-yl...)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296990(CHEMBL559348 | N-(5-Methanesulfonylamino-4,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297023(CHEMBL556232 | N-(1-Butyl-5-methanesulfonylamino-4...)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297019(CHEMBL551410 | N-[5-Methanesulfonylamino-1-(2-meth...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50263192(CHEMBL478858 | CHEMBL564483 | Pactimibe | [7-(2,2-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of ACAT-mediated esterified cholesterol accumulation in human THP1 cells exposed to acetyl-LDL after differentiation assessed as effect on...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1RX7PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297020(CHEMBL563918 | N-[1-(2-Ethoxyethyl)-5-methanesulfo...)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50263196(CHEMBL478015 | N-(5-Aminomethyl-4,6-dimethyl-1-oct...)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of ACAT-mediated esterified cholesterol accumulation in human THP1 cells exposed to acetyl-LDL during differentiation assessed as effect o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1RX7PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50209683((R)-2-(4-(9-bromo-2,3-dimethylnaphtho[2,3-b]thioph...)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297024(CHEMBL563699 | N-(1-Isobutyl-5-methanesulfonylamin...)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361277(CHEMBL1933093)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297004(CHEMBL554163 | N-(4,6-dimethyl-1-propylindolin-7-y...)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50263150(CHEMBL513892 | N-(4,6-dimethyl-1-octylindolin-7-yl...)copy SMILEScopy InChI
Affinity DataIC50: 640nMAssay Description:Inhibition of ACAT-mediated esterified cholesterol accumulation in human THP1 cells exposed to acetyl-LDL during differentiation assessed as effect o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1RX7PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296999(CHEMBL549714 | [1-Decyl-7-(2,2-dimethylpropanamido...)copy SMILEScopy InChI
Affinity DataIC50: 910nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361286(CHEMBL1935611)copy SMILEScopy InChI
Affinity DataIC50: 940nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361289(CHEMBL1935608)copy SMILEScopy InChI
Affinity DataIC50: 950nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297000(CHEMBL563263 | [7-(2,2-Dimethylpropanamido)-4,6-di...)copy SMILEScopy InChI
Affinity DataIC50: 960nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361293(CHEMBL1935501)copy SMILEScopy InChI
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361276(CHEMBL1935620)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361283(CHEMBL1935614)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297001(CHEMBL564069 | [7-(2,2-Dimethylpropanamido)-1-dode...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361292(CHEMBL1935607)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361287(CHEMBL1935610)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361295(CHEMBL1935499)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296998(CHEMBL558325 | [7-(2,2-Dimethylpropanamido)-4,6-di...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361298(CHEMBL1935496)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296989(CHEMBL561798 | N-(1-Ethyl-5-methanesulfonylamino-4...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TTCPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361296(CHEMBL1935498)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361294(CHEMBL1935500)copy SMILEScopy InChI
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361285(CHEMBL1935612)copy SMILEScopy InChI
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50069900(2,6-diisopropylphenyl 2-(2,4,6-triisopropylphenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of ACAT-mediated esterified cholesterol accumulation in human THP1 cells exposed to acetyl-LDL during differentiation assessed as effect o...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1RX7PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50361284(CHEMBL1935613)copy SMILEScopy InChI
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZZSPubMed
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