Compile Data Set for Download or QSAR
Found 54 with Last Name = 'matsuki' and Initial = 'k'
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035609(CHEMBL3338455)copy SMILEScopy InChI
Affinity DataIC50: 0.0530nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035620(CHEMBL3338445)copy SMILEScopy InChI
Affinity DataIC50: 0.130nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065697(CHEMBL3404016)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035617(CHEMBL3338448)copy SMILEScopy InChI
Affinity DataIC50: 0.380nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035621(CHEMBL3338444)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035613(CHEMBL3338452)copy SMILEScopy InChI
Affinity DataIC50: 0.740nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065689(CHEMBL3404009)copy SMILEScopy InChI
Affinity DataIC50: 0.860nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036633(CHEMBL3354285)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065686(CHEMBL3404006)copy SMILEScopy InChI
Affinity DataIC50: 0.980nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50100662(CHEMBL553371 | CHEMBL77971 | methyl 2-(4-aminophen...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PDE5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036625(CHEMBL3354279)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035618(CHEMBL3338447)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035611(CHEMBL3338453)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM14390(5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phen...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PDE5 (unknown origin)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065688(CHEMBL3404008)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035615(CHEMBL3338450)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035610(CHEMBL3338454)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036632(CHEMBL3354284)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035652(CHEMBL3338443)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036610(CHEMBL3354264)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035614(CHEMBL3338451)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036612(CHEMBL3354266)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065691(CHEMBL3404011)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065690(CHEMBL3404010)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035616(CHEMBL3338449)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036619(CHEMBL3354273)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035653(CHEMBL3338442)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036611(CHEMBL3354265)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035619(CHEMBL3338446)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036629(Avanafil | CHEBI:66876 | Stendra | TA-1790)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065695(CHEMBL3404014)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036609(CHEMBL3354287)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036616(CHEMBL3354270)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036634(CHEMBL3354286)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036624(CHEMBL3354278)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036631(CHEMBL3352836)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065687(CHEMBL3404007)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036618(CHEMBL3354272)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065692(CHEMBL3404012)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065694(CHEMBL3404013)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036613(CHEMBL3354267)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036617(CHEMBL3354271)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036615(CHEMBL3354269)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036628(CHEMBL3354282)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036621(CHEMBL3354275)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036620(CHEMBL3354274)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50065696(CHEMBL3404015)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP incubated for 30 mins by scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP54Z6PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50035654(CHEMBL3338441)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of canine lung PDE5 using [3H]cGMP substrate by radiolabeled nucleotide methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76F5ZPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036630(CHEMBL3354283)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50036623(CHEMBL3354277)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of dog lungs PDE5 using [3H]cGMP as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S1WPubMed
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