Compile Data Set for Download or QSAR
Found 104 with Last Name = 'mattia' and Initial = 'k'
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209260((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-methyl-N...)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209260((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-methyl-N...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Displacement of mouse MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209278((S)-N-(1-(2-carbamoylphenethyl)piperidin-4-yl)-1-(...)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209261((S)-N-(1-(2-fluorophenethyl)piperidin-4-yl)-1-(5-c...)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209251((S)-N-(1-(2-aminophenethyl)piperidin-4-yl)-1-(5-ch...)copy SMILEScopy InChI
Affinity DataKi:  280nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209257((S)-N-(1-(3-chlorophenethyl)piperidin-4-yl)-1-(5-c...)copy SMILEScopy InChI
Affinity DataKi:  400nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209279((S)-N-(1-(2-(trifluoromethyl)phenethyl)piperidin-4...)copy SMILEScopy InChI
Affinity DataKi:  420nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209262((S)-N-(1-(2-chlorophenethyl)piperidin-4-yl)-1-(5-c...)copy SMILEScopy InChI
Affinity DataKi:  460nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209265((S)-N-(1-(3-methoxyphenethyl)piperidin-4-yl)-1-(5-...)copy SMILEScopy InChI
Affinity DataKi:  470nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209260((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-methyl-N...)copy SMILEScopy InChI
Affinity DataKi:  500nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209253((S)-2-(2-(4-(1-(5-chloronaphthalen-2-ylsulfonyl)-N...)copy SMILEScopy InChI
Affinity DataKi:  530nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209268((S)-N-methyl-1-(naphthalen-2-ylsulfonyl)-N-(1-phen...)copy SMILEScopy InChI
Affinity DataKi:  590nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209255((S)-N-methyl-1-(naphthalen-2-ylsulfonyl)-N-(1-(3-p...)copy SMILEScopy InChI
Affinity DataKi:  620nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209258((S)-N-(1-(4-chlorophenethyl)piperidin-4-yl)-1-(5-c...)copy SMILEScopy InChI
Affinity DataKi:  820nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209269((S)-1-(5-fluoronaphthalen-2-ylsulfonyl)-N-methyl-N...)copy SMILEScopy InChI
Affinity DataKi:  850nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209263((S)-N-(1-benzylpiperidin-4-yl)-N-methyl-1-(naphtha...)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209281((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-ethyl-N-...)copy SMILEScopy InChI
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209270((S)-N-(1-benzylpiperidin-4-yl)-1-(naphthalen-2-yls...)copy SMILEScopy InChI
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209271((S)-2-(1-(naphthalen-2-ylsulfonyl)-N-(1-phenethylp...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209272((S)-1-(naphthalen-2-ylsulfonyl)-N-(1-(pyridin-2-yl...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209275((S)-N-(1-isobutylpiperidin-4-yl)-1-(naphthalen-2-y...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209256((S)-N-(1-benzylpiperidin-4-yl)-1-(4-isopropylpheny...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209252((S)-1-(5-chloronaphthalen-2-ylsulfonyl)-N-methyl-N...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209250((S)-N-methyl-1-(naphthalen-2-ylsulfonyl)-N-(1-(phe...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209247((S)-1-(5-aminonaphthalen-2-ylsulfonyl)-N-methyl-N-...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209273((S)-1-(5-acetamidonaphthalen-2-ylsulfonyl)-N-methy...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209246((S)-1-(naphthalen-2-ylsulfonyl)-N-(1-(pyridin-3-yl...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209248((S)-ethyl 2-(1-(naphthalen-2-ylsulfonyl)-N-(1-phen...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209274((S)-N-(2-morpholinoethyl)-1-(naphthalen-2-ylsulfon...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209249((S)-N-(1-benzylpiperidin-4-yl)-1-(benzylsulfonyl)p...)copy SMILEScopy InChI
Affinity DataKi:  1.50E+4nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209266((S)-N2-(1-benzylpiperidin-4-yl)-N1-(4-tert-butylph...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209277((R)-N-(1-benzylpiperidin-4-yl)-1-(naphthalen-2-yls...)copy SMILEScopy InChI
Affinity DataKi:  2.02E+4nMAssay Description:Displacement of human TARC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209276((S)-N-(1-benzylpiperidin-4-yl)-1-(naphthalen-2-ylm...)copy SMILEScopy InChI
Affinity DataKi:  2.50E+4nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209264((S)-N-(1-benzylpiperidin-4-yl)-N-methyl-1-(naphtha...)copy SMILEScopy InChI
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209259((S)-N-(1-benzylpiperidin-4-yl)-1-(phenylsulfonyl)p...)copy SMILEScopy InChI
Affinity DataKi: >2.90E+4nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209267((S)-1-(2-naphthoyl)-N-(1-benzylpiperidin-4-yl)pyrr...)copy SMILEScopy InChI
Affinity DataKi: >2.90E+4nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209280((S)-N-(1-benzylpiperidin-4-yl)-1-(isopropylsulfony...)copy SMILEScopy InChI
Affinity DataKi: >2.90E+4nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50209254((S)-1-(naphthalen-2-ylsulfonyl)-N-(piperidin-4-yl)...)copy SMILEScopy InChI
Affinity DataKi: >3.30E+4nMAssay Description:Displacement of human MDC from recombinant CCR4 receptor expressed in CHO cells coexpressing Galpha16 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9X2PPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129541(3-[5-(2',4'-Dichloro-biphenyl-4-yl)-3-tetrazol-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against Staphylococcus aureus methionyl-tRNA synthetase (SaMetRS)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129527(5-(2',4'-Dichloro-biphenyl-4-yl)-1-pyridin-3-yl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human methionyl-tRNA synthetase (hMetRS).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129528(2-[5-(2',4'-Dichloro-biphenyl-4-yl)-3-tetrazol-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against Staphylococcus aureus methionyl-tRNA synthetase (SaMetRS)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129551(CHEMBL74224 | {[5-(2',4'-Dichloro-biphenyl-4-yl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against Staphylococcus aureus methionyl-tRNA synthetase (SaMetRS)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129534(5-(2',4'-Dichloro-biphenyl-4-yl)-1-pyridin-3-yl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against human methionyl-tRNA synthetase (hMetRS).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129553(5-(2',4'-Dichloro-biphenyl-4-yl)-1-pyridin-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against Staphylococcus aureus methionyl-tRNA synthetase (SaMetRS)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129539(1-[5-(2',4'-Dichloro-biphenyl-4-yl)-1-(2-methoxy-p...)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibitory activity against Enterococci faecalis methionyl-tRNA synthetase (EfMetRS)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129546(5-(2',4'-Dichloro-biphenyl-4-yl)-1-pyridin-2-yl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibitory activity against human methionyl-tRNA synthetase (hMetRS).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129533(5-(2',4'-Dichloro-biphenyl-4-yl)-1-pyridin-3-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 660nMAssay Description:Inhibitory activity against Staphylococcus aureus methionyl-tRNA synthetase (SaMetRS)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129550(5-(2',4'-Dichloro-biphenyl-4-yl)-2-pyridin-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 910nMAssay Description:Inhibitory activity against Staphylococcus aureus methionyl-tRNA synthetase (SaMetRS)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129532(5-(2',4'-Dichloro-biphenyl-4-yl)-1-ethyl-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibitory activity against Staphylococcus aureus methionyl-tRNA synthetase (SaMetRS)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
TargetMethionine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Cubist Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50129543(5-(2',4'-Dichloro-biphenyl-4-yl)-2-pyridin-3-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibitory activity against human methionyl-tRNA synthetase (hMetRS).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7TCMPubMed
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