TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Inhibition of PGPH-like activity of 20S proteasome in human erythrocytes using Z-Leu-Leu-Glu-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Inhibition of bovine pancreatic alpha-chymotrypsin using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Inhibition of PGPH-like activity of 20S proteasome in human erythrocytes using Z-Leu-Leu-Glu-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 440nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 440nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 440nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 520nMAssay Description:Inhibition of human 20S proteasome post-glutamyl peptide hydrolyzing activity using Z-Leu-Leu-Glu-AMC as substrate measured over 10 mins by fluoresce...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 560nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 690nMAssay Description:Inhibition of PGPH-like activity of 20S proteasome in human erythrocytes using Z-Leu-Leu-Glu-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 990nMAssay Description:Inhibition of PGPH-like activity of 20S proteasome in human erythrocytes using Z-Leu-Leu-Glu-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.25E+3nMAssay Description:Inhibition of PGPH-like activity of 20S proteasome in human erythrocytes using Z-Leu-Leu-Glu-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.34E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.34E+3nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.38E+3nMAssay Description:Inhibition of human 20S proteasome post-glutamyl peptide hydrolyzing activity using Z-Leu-Leu-Glu-AMC as substrate measured over 10 mins by fluoresce...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.42E+3nMAssay Description:Inhibition of human 20S proteasome post-glutamyl peptide hydrolyzing activity using Z-Leu-Leu-Glu-AMC as substrate measured over 10 mins by fluoresce...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.45E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.45E+3nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.48E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.55E+3nMAssay Description:Inhibition of PGPH-like activity of 20S proteasome in human erythrocytes using Z-Leu-Leu-Glu-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.55E+3nMAssay Description:Inhibition of human 20S proteasome post-glutamyl peptide hydrolyzing activity using Z-Leu-Leu-Glu-AMC as substrate measured over 10 mins by fluoresce...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.62E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 1.62E+3nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 2.04E+3nMAssay Description:Inhibition of PGPH-like activity of 20S proteasome in human erythrocytes using Z-Leu-Leu-Glu-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 2.34E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of bovine pancreatic alpha-chymotrypsin using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 3.90E+3nMAssay Description:Inhibition of human 20S proteasome post-glutamyl peptide hydrolyzing activity using Z-Leu-Leu-Glu-AMC as substrate measured over 10 mins by fluoresce...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 4.42E+3nMAssay Description:Inhibition of human 20S proteasome post-glutamyl peptide hydrolyzing activity using Z-Leu-Leu-Glu-AMC as substrate measured over 10 mins by fluoresce...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 4.57E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataKi: 5.14E+3nMAssay Description:Inhibition of human 20S proteasome post-glutamyl peptide hydrolyzing activity using Z-Leu-Leu-Glu-AMC as substrate measured over 10 mins by fluoresce...More data for this Ligand-Target Pair