Compile Data Set for Download or QSAR
Found 62 with Last Name = 'seyb' and Initial = 'k'
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554754(CHEMBL4790764)copy SMILES
Affinity DataKi:  1.40nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554734(CHEMBL4761415 | US11530244, Compound 289)copy SMILES
Affinity DataKi:  1.5nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554755(CHEMBL4782157)copy SMILES
Affinity DataKi:  1.5nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554743(CHEMBL4759174)copy SMILES
Affinity DataKi:  2.10nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554736(CHEMBL4789838)copy SMILES
Affinity DataKi:  2.70nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554760(CHEMBL4798026)copy SMILES
Affinity DataKi:  2.80nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554735(CHEMBL4742833)copy SMILES
Affinity DataKi:  3.90nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554759(CHEMBL4745053)copy SMILES
Affinity DataKi:  4nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554731(CHEMBL4789480)copy SMILES
Affinity DataKi:  4nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554739(CHEMBL4789893)copy SMILES
Affinity DataKi:  4.20nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554750(CHEMBL4755930)copy SMILES
Affinity DataKi:  4.20nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554733(CHEMBL4754486)copy SMILES
Affinity DataKi:  4.20nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554732(CHEMBL4743963)copy SMILES
Affinity DataKi:  4.30nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554737(CHEMBL4776000)copy SMILES
Affinity DataKi:  6.30nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554753(CHEMBL4752664)copy SMILES
Affinity DataKi:  8.20nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554751(CHEMBL4794023)copy SMILES
Affinity DataKi:  9.40nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554749(CHEMBL4761848 | US11530244, Compound 461)copy SMILES
Affinity DataKi:  9.5nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554742(CHEMBL4760531)copy SMILES
Affinity DataKi:  10nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554741(CHEMBL4756076 | US11530244, Compound 042)copy SMILES
Affinity DataKi:  11nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554752(CHEMBL4743663 | US11530244, Compound 485)copy SMILES
Affinity DataKi:  11nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554756(CHEMBL4750201)copy SMILES
Affinity DataKi:  11nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554740(CHEMBL4795153 | US11530244, Compound 014)copy SMILES
Affinity DataKi:  12nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554744(CHEMBL4759663 | US11530244, Compound 248)copy SMILES
Affinity DataKi:  14nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554738(CHEMBL4783376)copy SMILES
Affinity DataKi:  23nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554745(CHEMBL4744423)copy SMILES
Affinity DataKi:  35nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554746(CHEMBL4797587)copy SMILES
Affinity DataKi:  39nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554758(CHEMBL4740923)copy SMILES
Affinity DataKi:  44nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554748(CHEMBL4761653 | US11530244, Compound 426)copy SMILES
Affinity DataKi:  81nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554747(CHEMBL4756880 | US11530244, Compound 425)copy SMILES
Affinity DataKi:  86nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554761(CHEMBL4759482)copy SMILES
Affinity DataKi:  175nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetProprotein convertase subtilisin/kexin type 9(Homo sapiens (Human))TBA
LigandPNGBDBM50554757(CHEMBL4779343)copy SMILES
Affinity DataKi:  285nMAssay Description:Inhibition of AlexaFluor647-tagged cyclic peptide binding to avi-tagged-biotinylated human PCSK9 measured after 2 hrs by Lance Streptavidin Europium ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N272NPubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311312(CHEMBL1078739 | N-(2-chlorophenyl)-6-phenylimidazo...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311306(CHEMBL1078214 | N-(2-chlorophenyl)-5-(piperidin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311302(CHEMBL1078107 | N-(2-chlorophenyl)-5-phenylpyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311303(CHEMBL1077571 | N-(2-chlorophenyl)-5-(dimethylamin...)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311316(CHEMBL1077739 | LDN-211904 | N-(2-chlorophenyl)-6-...)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311313(CHEMBL1078840 | N-(2-chlorophenyl)-6-(piperidin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311318(6-bromo-N-(2-chlorophenyl)-2-methylimidazo[1,2-a]p...)copy SMILEScopy InChI
Affinity DataIC50: 173nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311301(CHEMBL1080959 | N-(2-chlorophenyl)-5-methoxypyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311304(CHEMBL1078108 | N-(2-chlorophenyl)-5-(1H-pyrrol-1-...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311317(CHEMBL1077740 | N-(2-chlorophenyl)-6-(4-hydroxypip...)copy SMILEScopy InChI
Affinity DataIC50: 228nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311305(CHEMBL1078109 | N-(2-chlorophenyl)-5-morpholinopyr...)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311296(CHEMBL1081498 | N-(2-chlorophenyl)-5-methylpyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311311(CHEMBL1078738 | N-(2-chlorophenyl)imidazo[1,2-a]py...)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311288(CHEMBL1078785 | N-(2-chlorophenyl)pyrazolo[1,5-a]p...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311299(5-chloro-N-(2-chlorophenyl)pyrazolo[1,5-a]pyridine...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311297(CHEMBL1081499 | N-(2-chlorophenyl)-6-methylpyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311295(CHEMBL1080223 | N-(2-chlorophenyl)-4-methylpyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311310(CHEMBL1077850 | N-(2-chlorophenyl)pyrazolo[1,5-a]p...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
TargetEphrin type-B receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50311298(4-chloro-N-(2-chlorophenyl)pyrazolo[1,5-a]pyridine...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human recombinant EphB3 kinase-mediated BTK-peptide phosphorylation assessed as 33P incorporation after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43T66PubMed
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