Compile Data Set for Download or QSAR
Found 235 with Last Name = 'stenvall' and Initial = 'k'
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195247(CHEMBL3936580)copy SMILEScopy InChI
Affinity DataIC50: 0.251nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50011502(CHEMBL3261926)copy SMILEScopy InChI
Affinity DataIC50: 0.794nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195247(CHEMBL3936580)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195239(CHEMBL3972563 | US10287258, Example 29 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195239(CHEMBL3972563 | US10287258, Example 29 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280783(CHEMBL4164328)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280783(CHEMBL4164328)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of dihydrofolate reductase enzymes in Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195246(CHEMBL3980602 | US10287258, Example 16 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195246(CHEMBL3980602 | US10287258, Example 16 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195248(CHEMBL3891374 | US10287258, Example 27 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195248(CHEMBL3891374 | US10287258, Example 27 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195240(CHEMBL3960432 | US10287258, Example 3 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50011502(CHEMBL3261926)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195240(CHEMBL3960432 | US10287258, Example 3 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195238(CHEMBL3962926 | US10287258, Example 20 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280846(CHEMBL4171914)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Ability to inhibit HMG-CoA reductase (HMGR) by CoA reductase inhibition screen (COR) in ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280780(CHEMBL4169979)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280781(CHEMBL4164040)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280846(CHEMBL4171914)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Ability to inhibit HMG-CoA reductase (HMGR) by cholesterol synthesis inhibition screen (CSI) in ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195244(CHEMBL3926554 | US10287258, Example 24 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280848(CHEMBL4170481)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Ability to inhibit HMG-CoA reductase (HMGR) by CoA reductase inhibition screen (COR) in ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195238(CHEMBL3962926 | US10287258, Example 20 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195244(CHEMBL3926554 | US10287258, Example 24 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280780(CHEMBL4169979)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280781(CHEMBL4164040)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280848(CHEMBL4170481)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195245(CHEMBL3972158 | US10287258, Example 5 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195242(CHEMBL3917575 | US10287258, Example 14 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280852(CHEMBL4171040)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Ability to inhibit HMG-CoA reductase (HMGR) by cholesterol synthesis inhibition screen (CSI) in ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195242(CHEMBL3917575 | US10287258, Example 14 | US1066924...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Canis lupus familiaris)
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of dog DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280852(CHEMBL4171040)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195245(CHEMBL3972158 | US10287258, Example 5 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Rattus norvegicus)
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of rat DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50083974(2-Amino-N-[(R)-2-((R)-3a-benzyl-2-methyl-3-oxo-2,3...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50083974(2-Amino-N-[(R)-2-((R)-3a-benzyl-2-methyl-3-oxo-2,3...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of dihydrofolate reductase enzymes in Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195256(CHEMBL3954197)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Mus musculus)
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of mouse DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280785(CHEMBL4168863)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280785(CHEMBL4168863)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Ability to inhibit HMG-CoA reductase (HMGR) by CoA reductase inhibition screen (COR) in ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195236(CHEMBL3927609 | US10287258, Example 1 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195249(CHEMBL3970692)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280776(CHEMBL4174302)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Displacement of human [125I]-ghrelin from GHS-R1a (unknown origin) expressed in HEK293 cell membranes after 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50280776(CHEMBL4174302)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:In vitro inhibition of dihydrofolate reductase of Plasmodium bergheiMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD433XPubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195249(CHEMBL3970692)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195255(CHEMBL3945475 | US10287258, Example 6 | US10669245...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
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