TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]-3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:In vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:In vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:In vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:In vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro binding affinity at Dopamine receptor D2 of rat striatal membranes by [3H]-raclopride displacement.More data for this Ligand-Target Pair