Compile Data Set for Download or QSAR
Found 69 with Last Name = 'tomisawa' and Initial = 'k'
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50058163(Butyl-[2,5-dimethyl-7-(2,4,6-trimethyl-phenyl)-7H-...)copy SMILEScopy InChI
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50074456(CHEMBL10504 | SC241 | [3-(2-Bromo-4-isopropyl-phen...)copy SMILEScopy InChI
Affinity DataKi:  14.8nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85397(CRA1000)copy SMILEScopy InChI
Affinity DataKi:  15.7nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85398(CRA1001)copy SMILEScopy InChI
Affinity DataKi:  18.6nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85397(CRA1000)copy SMILEScopy InChI
Affinity DataKi:  20.6nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50074456(CHEMBL10504 | SC241 | [3-(2-Bromo-4-isopropyl-phen...)copy SMILEScopy InChI
Affinity DataKi:  20.7nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85398(CRA1001)copy SMILEScopy InChI
Affinity DataKi:  22.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50058163(Butyl-[2,5-dimethyl-7-(2,4,6-trimethyl-phenyl)-7H-...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85398(CRA1001)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50074456(CHEMBL10504 | SC241 | [3-(2-Bromo-4-isopropyl-phen...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85397(CRA1000)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GM85VGPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50170660(CHEMBL190883 | CHEMBL521582 | N,N-dipropyl-2-[4-me...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081380(CHEMBL553962 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081366(CHEMBL540331 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081369(CHEMBL128860 | CHEMBL541091 | [1-(4-Methoxy-3-phen...)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081371(CHEMBL128799 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081375(CHEMBL128717 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081372(CHEMBL127899 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081367(CHEMBL339638 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081376(CHEMBL341003 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 9.5nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081383(CHEMBL545760 | [2-(4-Methoxy-3-phenethyloxy-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081393(CHEMBL127720 | [2-(4-Methoxy-3-phenethyloxy-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081373(CHEMBL421446 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081370(CHEMBL340587 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081392(CHEMBL542470 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]-3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50074857(CHEMBL542786 | [2-(4-Methoxy-3-phenethyloxy-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50170660(CHEMBL190883 | CHEMBL521582 | N,N-dipropyl-2-[4-me...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:In vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081380(CHEMBL553962 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081385(1-(4-Methoxy-3-phenethyloxy-benzyl)-hexylamine; hy...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50074855(1-[2-(4-Methoxy-3-phenethyloxy-phenyl)-ethyl]-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081378(1-(4-Methoxy-3-phenethyloxy-benzyl)-4-methyl-penty...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081384(CHEMBL340275 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081377(1-(4-Methoxy-3-phenethyloxy-benzyl)-pentylamine | ...)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081388(1-(4-Methoxy-3-phenethyloxy-benzyl)-heptylamine | ...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081391(CHEMBL128999 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081366(CHEMBL540331 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:In vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081366(CHEMBL540331 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:In vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081366(CHEMBL540331 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081369(CHEMBL128860 | CHEMBL541091 | [1-(4-Methoxy-3-phen...)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:In vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081367(CHEMBL339638 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081389(CHEMBL128944 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081369(CHEMBL128860 | CHEMBL541091 | [1-(4-Methoxy-3-phen...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081371(CHEMBL128799 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081369(CHEMBL128860 | CHEMBL541091 | [1-(4-Methoxy-3-phen...)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081386(1-(4-Methoxy-3-phenethyloxy-benzyl)-butylamine; hy...)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081372(CHEMBL127899 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081375(CHEMBL128717 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081390(1-(4-Methoxy-3-phenethyloxy-benzyl)-octylamine | C...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50081376(CHEMBL341003 | [1-(4-Methoxy-3-phenethyloxy-benzyl...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:TIn vitro binding affinity at Sigma opioid receptor type 2 on guinea pig brain membranes by [3H]DTG displacement in the presence of [3H]pentazocine.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Taisho Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50170660(CHEMBL190883 | CHEMBL521582 | N,N-dipropyl-2-[4-me...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro binding affinity at Dopamine receptor D2 of rat striatal membranes by [3H]-raclopride displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7WQ7PubMed
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