Compile Data Set for Download or QSAR
Found 452 with Last Name = 'petrov' and Initial = 'kg'
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086433(CHEMBL3426034)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Inhibition of wild type fully glycosylated human recombinant CD38-catalyzed NAD hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086438(CHEMBL3426039)copy SMILEScopy InChI
Affinity DataKi:  0.450nMAssay Description:Inhibition of wild type fully glycosylated human recombinant CD38-catalyzed NAD hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086434(CHEMBL3426035)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Inhibition of wild type fully glycosylated human recombinant CD38-catalyzed NAD hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086425(CHEMBL3426030)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Inhibition of wild type fully glycosylated human recombinant CD38-catalyzed NAD hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086336(CHEMBL3426065)copy SMILES
Affinity DataIC50: 0.180nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086432(CHEMBL3426033)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086436(CHEMBL3426037)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086334(CHEMBL3426067)copy SMILEScopy InChI
Affinity DataIC50: 0.780nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086337(CHEMBL3426064)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086350(CHEMBL3426058)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256016(CHEMBL475768 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086335(CHEMBL3426066)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086431(CHEMBL3426032)copy SMILES
Affinity DataIC50: 1.30nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086438(CHEMBL3426039)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086336(CHEMBL3426065)copy SMILES
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086437(CHEMBL3426038)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086434(CHEMBL3426035)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086433(CHEMBL3426034)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256032(CHEMBL475594 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50142026(3-((1-methyl-1H-indol-3-yl)methylene)-1H-pyrrolo[3...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of receptor Tyrosine kinase A, TrkA (nerve growth factor receptor)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TDFPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086439(CHEMBL3426040)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256034((5-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)t...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256035(2-((5-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamin...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256036(CHEMBL474431 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086337(CHEMBL3426064)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086436(CHEMBL3426037)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086432(CHEMBL3426033)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086355(CHEMBL3426053)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256038(CHEMBL473437 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086351(CHEMBL3426057)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256017(CHEMBL475769 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086424(CHEMBL3426029)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086335(CHEMBL3426066)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256033(CHEMBL475761 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086435(CHEMBL3426036)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086334(CHEMBL3426067)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086431(CHEMBL3426032)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086430(CHEMBL3426031)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256039(CHEMBL473438 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50366932(CHEMBL1794058)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of receptor Tyrosine kinase A, TrkA (nerve growth factor receptor)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TDFPubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50142023(3-(5-Hydroxy-indan-1-ylidene)-1,3-dihydro-indol-2-...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of receptor Tyrosine kinase A, TrkA (nerve growth factor receptor)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TDFPubMed
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50576323(CHEMBL4866146)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of human HPGDS assessed as reduction in PGD2 formation using PGH2 as substrate by mass spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B28047PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256040(CHEMBL480349 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086333(CHEMBL3426027)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM27973(6-Ethynylthieno[3,2-d]pyrimidine, 8 | N-{3-chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 7nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7M35PubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50366929(CHEMBL1794057)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of receptor Tyrosine kinase A, TrkA (nerve growth factor receptor)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0TDFPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086324(CHEMBL3426186)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256020(CHEMBL475446 | N-(3-chloro-4-(3-fluorobenzyloxy)ph...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8NNNPubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086343(CHEMBL3426063)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of mouse recombinant CD38 extracellular domain expressed in CHO CGE cells assessed as NAD hydrolysis by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50086433(CHEMBL3426034)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9M00PubMed
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