TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 1.81E+3nMAssay Description:Binding affinity to human RXRalpha LBD after 15 mins by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2J38VDCPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2J38VDCPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 9nMAssay Description:Binding affinity to human RXRalpha LBD by fluorescence quenching methodMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 1.33E+3nMAssay Description:Binding affinity to human RXRalpha LBD after 15 mins by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 1.21E+3nMAssay Description:Binding affinity to human RXRalpha LBD after 15 mins by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 470nMAssay Description:Binding affinity to human RXRalpha LBD after 15 mins by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataEC50: 215nMAssay Description:Agonist activity at human RXRalpha LBD expressed in HEK293 cells transfected with Gal4 reporter assessed as increase of transcription by dual lucifer...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Agonist activity at human RXRalpha LBD expressed in HEK293 cells transfected with Gal4 reporter assessed as increase of transcription by dual lucifer...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Agonist activity at human RXRalpha LBD expressed in HEK293 cells transfected with Gal4 reporter assessed as increase of transcription by dual lucifer...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataEC50: 22nMAssay Description:Agonist activity at human RXRalpha LBD expressed in HEK293 cells transfected with Gal4 reporter assessed as increase of transcription by dual lucifer...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at human RXRalpha LBD expressed in HEK293 cells transfected with Gal4 reporter assessed as increase of transcription by dual lucifer...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataEC50: 118nMAssay Description:Agonist activity at RXRalpha LBD (unknown origin) expressed in CV1 cellsMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2J38VDCPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2J38VDCPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at human RXRalpha LBD expressed in HEK293 cells transfected with Gal4 reporter assessed as increase of transcription by dual lucifer...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at human RXRalpha LBD expressed in HEK293 cells transfected with Gal4 reporter assessed as increase of transcription by dual lucifer...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding affinity to human RXRalpha LBD by fluorescence quenching methodMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 9nMAssay Description:Binding affinity to human RXRalpha LBD by fluorescence quenching methodMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 35nMAssay Description:Binding affinity to human RXRalpha LBD by fluorescence quenching methodMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Binding affinity to human RXRalpha LBD by fluorescence quenching methodMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 125nMAssay Description:Binding affinity to human RXRalpha LBD by fluorescence quenching methodMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 34nMAssay Description:Binding affinity to human RXRalpha LBD by fluorescence quenching methodMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Alabama at Birmingham
Curated by ChEMBL
University of Alabama at Birmingham
Curated by ChEMBL
Affinity DataKd: 1.59E+3nMAssay Description:Binding affinity to human RXRalpha LBD after 15 mins by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2J38VDCPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2J38VDCPubMedDrugBank
MMDB
PDB
3D Structure (crystal)