Compile Data Set for Download or QSAR
Found 87 with Last Name = 'liu' and Initial = 'kl'
TargetPolycomb protein EED(Homo sapiens (Human))TBA
LigandPNGBDBM50609343(CHEMBL5269445)copy SMILES
Affinity DataIC50: 4.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583904(CHEMBL5091313)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
LigandPNGBDBM50241662(CHEMBL4104741)copy SMILEScopy InChI
Affinity DataIC50: 18nMMore data for this Ligand-Target Pair
In DepthDetails
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant N-terminal 6his-tagged BRD4 expressed in Escherichia coli BL21(DE3) using H4 peptide as substrate by alphascreen assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583911(CHEMBL5079375)copy SMILES
Affinity DataIC50: 40nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583914(CHEMBL5074971)copy SMILES
Affinity DataIC50: 50nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583906(CHEMBL5075342)copy SMILES
Affinity DataIC50: 100nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583902(CHEMBL5091281)copy SMILES
Affinity DataIC50: 180nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583898(CHEMBL5084409)copy SMILES
Affinity DataIC50: 180nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of BRD4 bromodomain (unknown origin)More data for this Ligand-Target Pair
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583900(CHEMBL5090481)copy SMILES
Affinity DataIC50: 320nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetPolycomb protein EED(Homo sapiens (Human))TBA
LigandPNGBDBM50236003(CHEMBL4096234)copy SMILEScopy InChI
Affinity DataIC50: 320nMMore data for this Ligand-Target Pair
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583895(CHEMBL5078063)copy SMILES
Affinity DataIC50: 330nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant N-terminal 6his-tagged BRD4 bromodomain 2 expressed in Escherichia coli BL21(DE3) using using H4 peptide as substrate...More data for this Ligand-Target Pair
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583915(CHEMBL5091279)copy SMILES
Affinity DataIC50: 530nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525654(CHEMBL4533819)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583889(CHEMBL5070084)copy SMILES
Affinity DataIC50: 560nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583908(CHEMBL5081296)copy SMILES
Affinity DataIC50: 640nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525650(CHEMBL4592461)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525648(CHEMBL4471181)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetPolycomb protein EED(Homo sapiens (Human))TBA
LigandPNGBDBM50259910(CHEMBL4097892)copy SMILEScopy InChI
Affinity DataIC50: 890nMMore data for this Ligand-Target Pair
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583899(CHEMBL5075319)copy SMILES
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525657(CHEMBL4581142)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525647(CHEMBL4456714)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetPolycomb protein EED(Homo sapiens (Human))TBA
LigandPNGBDBM223984(rac-(3R,4S)-1-(2-methoxybenzyl)-N,N-dimethyl-4-(1-...)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525656(CHEMBL4527844)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525649(CHEMBL4555713)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50216786(CHEMBL229457 | N-(7-Amino-heptyl)-guanidine | N-gu...)copy SMILEScopy InChI
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525655(CHEMBL4460102)copy SMILEScopy InChI
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525652(CHEMBL4472855)copy SMILEScopy InChI
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525653(CHEMBL4461915)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525646(CHEMBL4582953)copy SMILEScopy InChI
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525651(CHEMBL4470171)copy SMILEScopy InChI
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583888(CHEMBL5089864)copy SMILES
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583894(CHEMBL5080635)copy SMILES
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525658(CHEMBL4574735)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P13FZPubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583891(CHEMBL5080971)copy SMILES
Affinity DataIC50: 4.31E+3nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583893(CHEMBL5073964)copy SMILES
Affinity DataIC50: 4.42E+3nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583896(CHEMBL5078229)copy SMILES
Affinity DataIC50: 5.43E+3nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetPolycomb protein EED(Homo sapiens (Human))TBA
LigandPNGBDBM50609344(CHEMBL5273243)copy SMILES
Affinity DataIC50: 8.76E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetPolycomb protein EED(Homo sapiens (Human))TBA
LigandPNGBDBM50410562(CHEMBL5269781)copy SMILEScopy InChI
Affinity DataIC50: 1.16E+4nMMore data for this Ligand-Target Pair
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583890(CHEMBL5091549)copy SMILES
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583909(CHEMBL5081865)copy SMILES
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583910(CHEMBL5092133)copy SMILES
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583907(CHEMBL5089522)copy SMILES
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50570077(CHEMBL4874971)copy SMILES
Affinity DataIC50: 2.64E+4nMAssay Description:Inhibition of recombinant human His-tagged VEGFR2 expressed in Baculovirus expression system using ADP-Glo as substrate measured after 30 mins in pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K4BPubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583913(CHEMBL5069826)copy SMILES
Affinity DataIC50: 3.37E+4nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50583905(CHEMBL5072102)copy SMILES
Affinity DataIC50: 3.58E+4nMAssay Description:Inhibition of DHPS (unknown origin ) incubated for 30 mins by NAD/NADH-Glow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MH5PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50570091(CHEMBL4866291)copy SMILES
Affinity DataIC50: 3.69E+4nMAssay Description:Inhibition of recombinant human His-tagged VEGFR2 expressed in Baculovirus expression system using ADP-Glo as substrate measured after 30 mins in pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K4BPubMed
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