Compile Data Set for Download or QSAR
Found 96 with Last Name = 'stark' and Initial = 'kl'
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059194(CHEMBL3393337)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059190(CHEMBL3393333)copy SMILEScopy InChI
Affinity DataKi: <0.5nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059191(CHEMBL3393334)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059201(CHEMBL3393329)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059202(CHEMBL3393327)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059198(CHEMBL3393340)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059205(CHEMBL3393322 | US9868720, No. 92)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059211(CHEMBL3393314)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059189(CHEMBL3393332)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059200(CHEMBL3393330)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059207(CHEMBL3393320)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059206(CHEMBL3393321)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059193(CHEMBL3393336)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059192(CHEMBL3393335)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059199(CHEMBL3393331)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059197(CHEMBL3393339)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059210(CHEMBL3393315)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059212(CHEMBL3393312)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059215(CHEMBL3393328)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059203(CHEMBL3393324)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059214(CHEMBL3393308)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059204(CHEMBL3393323)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059208(CHEMBL3393318)copy SMILEScopy InChI
Affinity DataKi:  57nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059213(CHEMBL3393310)copy SMILEScopy InChI
Affinity DataKi:  85nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059209(CHEMBL3393317)copy SMILEScopy InChI
Affinity DataKi:  90nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059196(CHEMBL3393338)copy SMILEScopy InChI
Affinity DataKi:  93nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059226(CHEMBL3393325)copy SMILEScopy InChI
Affinity DataKi:  166nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059249(CHEMBL3393313 | US9868720, No. 6)copy SMILEScopy InChI
Affinity DataKi:  195nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059257(CHEMBL3393309 | US9868720, No. 5)copy SMILEScopy InChI
Affinity DataKi:  401nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059216(CHEMBL3393326)copy SMILEScopy InChI
Affinity DataKi:  431nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059253(CHEMBL3393311 | US9868720, No. 3)copy SMILEScopy InChI
Affinity DataKi:  691nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059244(CHEMBL3393319)copy SMILEScopy InChI
Affinity DataKi:  725nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059248(CHEMBL3393316)copy SMILEScopy InChI
Affinity DataKi:  942nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059190(CHEMBL3393333)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50122512(3-{4-[2-(4-Fluoro-phenyl)-2-(4-methyl-piperazin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:In vitro ability to inhibit the binding of [125I]-AGRP to the human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZQ1PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059191(CHEMBL3393334)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059198(CHEMBL3393340)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059194(CHEMBL3393337)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059190(CHEMBL3393333)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059202(CHEMBL3393327)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059201(CHEMBL3393329)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059200(CHEMBL3393330)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059207(CHEMBL3393320)copy SMILEScopy InChI
Affinity DataIC50: 109nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50122513(1-(4-Chloro-phenyl)-3-{4-[2-(4-chloro-phenyl)-2-(4...)copy SMILEScopy InChI
Affinity DataIC50: 118nMAssay Description:In vitro ability to inhibit the binding of [125I]-AGRP to the human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZQ1PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059189(CHEMBL3393332)copy SMILEScopy InChI
Affinity DataIC50: 125nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059190(CHEMBL3393333)copy SMILEScopy InChI
Affinity DataIC50: 129nMAssay Description:Inhibition of JNK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50059193(CHEMBL3393336)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50122513(1-(4-Chloro-phenyl)-3-{4-[2-(4-chloro-phenyl)-2-(4...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:In vitro ability to inhibit the binding of alpha [125I]-NDP-MSH to the human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZQ1PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50122508(3-{4-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-fluoro-...)copy SMILEScopy InChI
Affinity DataIC50: 152nMAssay Description:In vitro ability to inhibit the binding of [125I]-AGRP to the human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZQ1PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50122508(3-{4-[2-(4-Cyclohexyl-piperazin-1-yl)-2-(4-fluoro-...)copy SMILEScopy InChI
Affinity DataIC50: 164nMAssay Description:In vitro ability to inhibit the binding of alpha [125I]-NDP-MSH to the human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZQ1PubMed
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