TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of methionine aminopeptidase 2More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of HSP90 (unknown origin)More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of methionine aminopeptidase 2More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2SN0CG4PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2SN0CG4PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
Affinity DataIC50: 700nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of methionine aminopeptidase 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of methionine aminopeptidase 1More data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2765G84PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2765G84PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of methionine aminopeptidase 1More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of methionine aminopeptidase 2More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.77E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of methionine aminopeptidase 2More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of methionine aminopeptidase 2More data for this Ligand-Target Pair
![](/img/powered_by_small.gif)