Compile Data Set for Download or QSAR
Found 353 with Last Name = '?rfi' and Initial = 'l'
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454441(CHEMBL4217448)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454379(CHEMBL4205123)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454411(CHEMBL4209151)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human partial length FLT3 ITD mutant expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50277584(CHEMBL482968 | N-(5-methyl-1H-pyrazol-3-yl)-6-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454382(CHEMBL4206688)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50504574(CHEMBL4469622)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of FLT3 (unknown origin) autophosphorylation expressed in BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454399(CHEMBL4215419)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454410(CHEMBL4212641)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454396(CHEMBL4207754)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454402(CHEMBL4209357)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454392(CHEMBL4204526)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454453(CHEMBL4211020)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454384(CHEMBL4205779)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454397(CHEMBL4215514)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454387(CHEMBL4216304)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454383(CHEMBL4206359)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of wild-type human partial length FLT3 (V592 to Y969 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454386(CHEMBL4205084)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467014(CHEMBL4279747)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454404(CHEMBL4209987)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454385(CHEMBL4218213)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454456(CHEMBL4213505)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50355496(CHEMBL1908397)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human FLT3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454395(CHEMBL4203989)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454393(CHEMBL4216190)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454445(CHEMBL4203392)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467013(CHEMBL4290876)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454457(CHEMBL4203224)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454440(CHEMBL4217685)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454403(CHEMBL4210799)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50277584(CHEMBL482968 | N-(5-methyl-1H-pyrazol-3-yl)-6-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human GST-tagged PDGFR alpha (550 to 1089 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50277584(CHEMBL482968 | N-(5-methyl-1H-pyrazol-3-yl)-6-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human full length His-tagged Src expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50277584(CHEMBL482968 | N-(5-methyl-1H-pyrazol-3-yl)-6-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human His-tagged FMS expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50277584(CHEMBL482968 | N-(5-methyl-1H-pyrazol-3-yl)-6-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human GST-tagged RET expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50277584(CHEMBL482968 | N-(5-methyl-1H-pyrazol-3-yl)-6-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human His-tagged VEGFR 2 expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50177716(CHEMBL3813873 | US11679110, Compound Pexidartinib ...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454389(CHEMBL4216726)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467019(CHEMBL4277642)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454394(CHEMBL4205921)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454401(CHEMBL4202527)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454390(CHEMBL4215592)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd

Curated by ChEMBL
LigandPNGBDBM50177716(CHEMBL3813873 | US11679110, Compound Pexidartinib ...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant FMS (unknown origin)More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50277584(CHEMBL482968 | N-(5-methyl-1H-pyrazol-3-yl)-6-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant full length His-tagged human aurora A using peptide substrate in presence of ATP at its Km concentration by Z-lyte kinase a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27947ZVPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454449(CHEMBL4211337)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.

Curated by ChEMBL
LigandPNGBDBM50517975(CHEMBL4589698)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077NZPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467014(CHEMBL4279747)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50454391(CHEMBL4204994)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867XNPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.

Curated by ChEMBL
LigandPNGBDBM50518002(CHEMBL4439964)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077NZPubMed
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