Compile Data Set for Download or QSAR
Found 63 with Last Name = 'bayless' and Initial = 'l'
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50073179(8-Chloro-11-piperidin-4-ylidene-6,11-dihydro-5H-be...)copy SMILEScopy InChI
Affinity DataKi:  0.970nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMedDrugBank
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155336(1-{4-[4-(4-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataKi:  3.63nMAssay Description:Binding affinity for recombinant human Histamine H1 receptor expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144624((5-{4-[(R)-(4-Chloro-phenyl)-phenyl-methyl]-pipera...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:In vitro binding affinity towards histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160828(CHEMBL366925 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataKi:  5.01nMAssay Description:Binding affinity for human Histamine H1 receptor in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM22890(2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-...)copy SMILEScopy InChI
Affinity DataKi:  5.89nMAssay Description:Binding affinity for human Histamine H1 receptor in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMedDrugBank
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160827(CHEMBL179590 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataKi:  5.89nMAssay Description:Binding affinity for human Histamine H1 receptor in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160831(CHEMBL181085 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataKi:  7.59nMAssay Description:Binding affinity for human Histamine H1 receptor in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155335(1-{4-[4-(3-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]...)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160829(CHEMBL180233 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataKi:  9.55nMAssay Description:Binding affinity for human Histamine H1 receptor in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155341(1-(4-{4-[3-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM22890(2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMedDrugBank
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM22890(2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:In vitro binding affinity towards histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMedDrugBank
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160830(CHEMBL360666 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataKi:  17.8nMAssay Description:Binding affinity for human Histamine H1 receptor in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155337(1-(4-{4-[2-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,...)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155336(1-{4-[4-(4-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155338(1-{4-[4-(4-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155334(1-(4-{4-[4-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,...)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144626(CHEMBL305662 | [4-((2S,5S)-5-{4-[(R)-(4-Chloro-phe...)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:In vitro binding affinity towards histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155339(1-{4-[4-(3-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataKi:  109nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144625(1-[4-(5-{4-[(R)-(4-Chloro-phenyl)-phenyl-methyl]-p...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:In vitro binding affinity towards histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144627(CHEMBL74688 | [4-((2R,5R)-5-{4-[(R)-(4-Chloro-phen...)copy SMILEScopy InChI
Affinity DataKi:  180nMAssay Description:In vitro binding affinity towards histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144622(CHEMBL312082 | [3-(5-{4-[(R)-(4-Chloro-phenyl)-phe...)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:In vitro binding affinity towards histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155340(1-{4-[4-(2-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataKi:  295nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155333(1-{4-[4-(2-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]...)copy SMILEScopy InChI
Affinity DataKi:  305nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM22876(CHEMBL998 | Claritin | Loratadine | Sch 29851 | US...)copy SMILEScopy InChI
Affinity DataKi:  414nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMedDrugBank
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144620(CHEMBL73706 | [4-(5-{4-[Bis-(4-fluoro-phenyl)-meth...)copy SMILEScopy InChI
Affinity DataKi:  550nMAssay Description:In vitro binding affinity towards histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144623(CHEMBL74779 | [4-((2S,5S)-5-{4-[Bis-(4-fluoro-phen...)copy SMILEScopy InChI
Affinity DataKi:  660nMAssay Description:In vitro binding affinity towards histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155340(1-{4-[4-(2-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155334(1-(4-{4-[4-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,...)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155338(1-{4-[4-(4-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]...)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160827(CHEMBL179590 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibitory concentration against 5-lipoxygenase in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155336(1-{4-[4-(4-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155336(1-{4-[4-(4-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Inhibitory concentration against 5-lipoxygenase in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155339(1-{4-[4-(3-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160828(CHEMBL366925 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibitory concentration against 5-lipoxygenase in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155335(1-{4-[4-(3-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]...)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160829(CHEMBL180233 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataIC50: 102nMAssay Description:Inhibitory concentration against 5-lipoxygenase in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144621(CHEMBL73148 | CMI-977 | N-(4-{(2S,5S)-5-[(4-fluoro...)copy SMILEScopy InChI
Affinity DataIC50: 117nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase in a human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144623(CHEMBL74779 | [4-((2S,5S)-5-{4-[Bis-(4-fluoro-phen...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase in a human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160830(CHEMBL360666 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibitory concentration against 5-lipoxygenase in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50029781((R)-(+)-N-{3-[5-(4-fluorobenzyl)thien-2-yl]-1-meth...)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase in a human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160828(CHEMBL366925 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibitory concentration against human 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144620(CHEMBL73706 | [4-(5-{4-[Bis-(4-fluoro-phenyl)-meth...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase in a human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50160831(CHEMBL181085 | N-hydroxycarbamate derivative)copy SMILEScopy InChI
Affinity DataIC50: 176nMAssay Description:Inhibitory concentration against 5-lipoxygenase in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155337(1-(4-{4-[2-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,...)copy SMILEScopy InChI
Affinity DataIC50: 185nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155336(1-{4-[4-(4-{4-[bis(4-fluorophenyl)methyl]piperazin...)copy SMILEScopy InChI
Affinity DataIC50: 193nMAssay Description:Inhibitory concentration against human 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN954NPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155341(1-(4-{4-[3-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,...)copy SMILEScopy InChI
Affinity DataIC50: 194nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144620(CHEMBL73706 | [4-(5-{4-[Bis-(4-fluoro-phenyl)-meth...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase in an RBL-2H3 cell lysateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
UCB Research

Curated by ChEMBL
LigandPNGBDBM50144625(1-[4-(5-{4-[(R)-(4-Chloro-phenyl)-phenyl-methyl]-p...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase in an RBL-2H3 cell lysateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7G2PPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
UCB Research

Curated by ChEMBL
LigandPNGBDBM50155333(1-{4-[4-(2-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]...)copy SMILEScopy InChI
Affinity DataIC50: 213nMAssay Description:Inhibition of 5-lipooxygenase activity in human whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9VRHPubMed
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