TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences, Inc.
Curated by PDSP Ki Database
Affinity DataIC50: 2.40nMAssay Description:Binding affinity towards Nicotinic acetylcholine receptor by the displacement of [3H]-nicotine from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Binding affinity towards Nicotinic acetylcholine receptor by the displacement of [3H]-nicotine from rat cortical membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataIC50: 1.60E+3nMAssay Description:The compound was tested on recombinant human alpha4-beta2 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataIC50: 4.50E+3nMAssay Description:The compound was tested on recombinant human alpha4-beta4 cell lines of HUman embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataIC50: 5.80E+3nMAssay Description:The compound was tested on recombinant human alpha2-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataIC50: 8.90E+3nMAssay Description:The compound was tested on recombinant human alpha3-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataIC50: 1.01E+4nMAssay Description:The compound was tested on recombinant human alpha3-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataIC50: 3.60E+5nMAssay Description:The compound was tested on recombinant human alpha3-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 1.50E+4nMAssay Description:The compound was tested on recombinant human alpha4-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 1.50E+4nMAssay Description:Binding affinity at NAChRs was determined by measuring the displacement of ([3H]Nic) from a preparation of rat cortical membranes.More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 2.90E+4nMAssay Description:Binding affinity at NAChRs was determined by measuring the displacement of ([3H]Nic) from a preparation of rat cortical membranes.More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit delta(Torpedo californica)
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 3.10E+4nMAssay Description:The compound was tested on recombinant human alpha3-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 5.10E+4nMAssay Description:The compound was tested on recombinant human alpha2-beta4 cell lines of HUman embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 5.00E+3nMAssay Description:The compound was tested on recombinant human alpha2-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 5.00E+3nMAssay Description:The compound was tested on recombinant human alpha2-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+4nMAssay Description:The compound was tested on recombinant human alpha2-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 4.10E+4nMAssay Description:The compound was tested on recombinant human alpha3-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 4.10E+4nMAssay Description:The compound was tested on recombinant human alpha3-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 9.00E+3nMAssay Description:The compound was tested on recombinant human alpha4-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 9.00E+3nMAssay Description:The compound was tested on recombinant human alpha4-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 2.30E+4nMAssay Description:The compound was tested on recombinant human alpha3-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 2.30E+4nMAssay Description:The compound was tested on recombinant human alpha3-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 2.60E+3nMAssay Description:The compound was tested on recombinant human alpha4-beta2 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 2.60E+3nMAssay Description:The compound was tested on recombinant human alpha4-beta2 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 2.30E+4nMAssay Description:The compound was tested on recombinant human alpha4-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 2.50E+4nMAssay Description:The compound was tested on recombinant human alpha4-beta4 cell lines of Human embryonic kidney for nicotinic acetylcholine receptor agonist functiona...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Homo sapiens (Human))
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
SIBIA Neurosciences Inc.
Curated by PDSP Ki Database
Affinity DataEC50: 3.20E+4nMAssay Description:Compound was evaluated for its agonist activity against activated human recombinant Nicotinic acetylcholine receptor alpha4-beta4 in Xenopus OocytesMore data for this Ligand-Target Pair
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