Compile Data Set for Download or QSAR
Found 25 with Last Name = 'fleury' and Initial = 'l'
TargetCeramide transfer protein(Homo sapiens (Human))
Universit£ Paul Sabatier-Toulouse III

Curated by ChEMBL
LigandPNGBDBM50067350(CHEMBL3401790)copy SMILEScopy InChI
Affinity DataEC50:  2.50E+4nMAssay Description:Binding affinity to histidine-tagged human recombinant COL4A3ABP containing CERT START domain pre-incubated for 30 mins before biotinylated ceramide ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5PVMPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239289(CHEMBL4096752)copy SMILEScopy InChI
Affinity DataEC50:  2.70E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetCeramide transfer protein(Homo sapiens (Human))
Universit£ Paul Sabatier-Toulouse III

Curated by ChEMBL
LigandPNGBDBM50067352(CHEMBL122892)copy SMILEScopy InChI
Affinity DataEC50:  2.20E+4nMAssay Description:Binding affinity to histidine-tagged human recombinant COL4A3ABP containing CERT START domain pre-incubated for 30 mins before biotinylated ceramide ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5PVMPubMed
TargetCeramide transfer protein(Homo sapiens (Human))
Universit£ Paul Sabatier-Toulouse III

Curated by ChEMBL
LigandPNGBDBM50067353(CHEMBL3401792)copy SMILEScopy InChI
Affinity DataEC50:  4.00E+3nMAssay Description:Binding affinity to histidine-tagged human recombinant COL4A3ABP containing CERT START domain pre-incubated for 30 mins before biotinylated ceramide ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5PVMPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239284(CHEMBL4096360)copy SMILEScopy InChI
Affinity DataEC50:  4.40E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239285(CHEMBL4096869)copy SMILEScopy InChI
Affinity DataEC50:  2.10E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239286(CHEMBL4084601)copy SMILEScopy InChI
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239287(CHEMBL4100095)copy SMILEScopy InChI
Affinity DataEC50:  6.80E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239288(CHEMBL4097685)copy SMILEScopy InChI
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239289(CHEMBL4096752)copy SMILEScopy InChI
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239290(CHEMBL4099197)copy SMILEScopy InChI
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239291(CHEMBL4091463)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239284(CHEMBL4096360)copy SMILEScopy InChI
Affinity DataEC50:  4.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239285(CHEMBL4096869)copy SMILEScopy InChI
Affinity DataEC50:  2.40E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239286(CHEMBL4084601)copy SMILEScopy InChI
Affinity DataEC50:  3.20E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239287(CHEMBL4100095)copy SMILEScopy InChI
Affinity DataEC50:  7.30E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239288(CHEMBL4097685)copy SMILEScopy InChI
Affinity DataEC50:  2.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239290(CHEMBL4099197)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+5nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239292(CHEMBL4070549)copy SMILEScopy InChI
Affinity DataEC50:  1.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239291(CHEMBL4091463)copy SMILEScopy InChI
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239293(CHEMBL4076088)copy SMILEScopy InChI
Affinity DataEC50:  1.40E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239294(CHEMBL4070517)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239292(CHEMBL4070549)copy SMILEScopy InChI
Affinity DataEC50:  1.90E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239293(CHEMBL4076088)copy SMILEScopy InChI
Affinity DataEC50:  3.00E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetCeramide transfer protein(Homo sapiens (Human))
Universit£ Paul Sabatier-Toulouse III

Curated by ChEMBL
LigandPNGBDBM50067351(CHEMBL3401791)copy SMILEScopy InChI
Affinity DataEC50:  1.59E+5nMAssay Description:Binding affinity to histidine-tagged human recombinant COL4A3ABP containing CERT START domain pre-incubated for 30 mins before biotinylated ceramide ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5PVMPubMed