Compile Data Set for Download or QSAR
Found 59 with Last Name = 'frankiewicz' and Initial = 'l'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070377(CHEMBL3408519)copy SMILEScopy InChI
Affinity DataKi:  0.0800nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155796(CHEMBL3781680)copy SMILEScopy InChI
Affinity DataKi:  0.187nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070377(CHEMBL3408519)copy SMILEScopy InChI
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50346329((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)copy SMILEScopy InChI
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50346329((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)copy SMILEScopy InChI
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155774(CHEMBL3780776)copy SMILEScopy InChI
Affinity DataKi:  0.990nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155794(CHEMBL3780820)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155798(CHEMBL3781519)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155795(CHEMBL3780408)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155799(CHEMBL3781336)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155798(CHEMBL3781519)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155799(CHEMBL3781336)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155800(CHEMBL3780686)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155797(CHEMBL3780818)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155800(CHEMBL3780686)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070377(CHEMBL3408519)copy SMILEScopy InChI
Affinity DataKi:  6.40nMAssay Description:Antagonist activity against human NK1 receptor expressed in CHO-K1 cells by aequorin luminescence assay based Schild's plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155800(CHEMBL3780686)copy SMILEScopy InChI
Affinity DataKi:  6.70nMAssay Description:Antagonist activity against human NK1 receptor expressed in CHO-K1 cells by aequorin luminescence assay based Schild's plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155800(CHEMBL3780686)copy SMILEScopy InChI
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155799(CHEMBL3781336)copy SMILEScopy InChI
Affinity DataKi:  7.5nMAssay Description:Antagonist activity against human NK1 receptor expressed in CHO-K1 cells by aequorin luminescence assay based Schild's plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50346329((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)copy SMILEScopy InChI
Affinity DataKi:  7.80nMAssay Description:Antagonist activity against human NK1 receptor expressed in CHO-K1 cells by aequorin luminescence assay based Schild's plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155798(CHEMBL3781519)copy SMILEScopy InChI
Affinity DataKi:  8.10nMAssay Description:Antagonist activity against human NK1 receptor expressed in CHO-K1 cells by aequorin luminescence assay based Schild's plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155797(CHEMBL3780818)copy SMILEScopy InChI
Affinity DataKi:  8.30nMAssay Description:Antagonist activity against human NK1 receptor expressed in CHO-K1 cells by aequorin luminescence assay based Schild's plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155774(CHEMBL3780776)copy SMILEScopy InChI
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50346329((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155799(CHEMBL3781336)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155798(CHEMBL3781519)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070377(CHEMBL3408519)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]SP from human NK1 receptor transfected in CHO cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155797(CHEMBL3780818)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155795(CHEMBL3780408)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155794(CHEMBL3780820)copy SMILEScopy InChI
Affinity DataKi:  54nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155796(CHEMBL3781680)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155795(CHEMBL3780408)copy SMILEScopy InChI
Affinity DataKi:  339nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155774(CHEMBL3780776)copy SMILEScopy InChI
Affinity DataKi:  533nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)copy SMILEScopy InChI
Affinity DataKi:  877nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155794(CHEMBL3780820)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155797(CHEMBL3780818)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070377(CHEMBL3408519)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070377(CHEMBL3408519)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155796(CHEMBL3781680)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155796(CHEMBL3781680)copy SMILEScopy InChI
Affinity DataIC50: 7.70nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50346329((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)copy SMILEScopy InChI
Affinity DataIC50: 8.5nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155800(CHEMBL3780686)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155799(CHEMBL3781336)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155799(CHEMBL3781336)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155798(CHEMBL3781519)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155798(CHEMBL3781519)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50155800(CHEMBL3780686)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QQJPubMed
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