Compile Data Set for Download or QSAR
Found 32 with Last Name = 'kindon' and Initial = 'l'
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50417257(SB-649868)copy SMILEScopy InChI
Affinity DataKi:  0.0776nMAssay Description:Antagonist activity at recombinant rat OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Rattus norvegicus (Rat))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50417257(SB-649868)copy SMILEScopy InChI
Affinity DataKi:  0.117nMAssay Description:Antagonist activity at recombinant rat OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419142(CHEMBL1830963)copy SMILEScopy InChI
Affinity DataKi:  0.126nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419136(CHEMBL1830961)copy SMILEScopy InChI
Affinity DataKi:  0.158nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419142(CHEMBL1830963)copy SMILEScopy InChI
Affinity DataKi:  0.251nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50417257(SB-649868)copy SMILEScopy InChI
Affinity DataKi:  0.316nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50417257(SB-649868)copy SMILEScopy InChI
Affinity DataKi:  0.398nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50417257(SB-649868)copy SMILEScopy InChI
Affinity DataKi:  0.759nMAssay Description:Displacement of [3H]almorexant from recombinant human OX1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419136(CHEMBL1830961)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419131(CHEMBL1830968)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50417257(SB-649868)copy SMILEScopy InChI
Affinity DataKi:  1.29nMAssay Description:Displacement of [3H]almorexant from recombinant human OX2R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419137(CHEMBL1830959)copy SMILEScopy InChI
Affinity DataKi:  5.01nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419131(CHEMBL1830968)copy SMILEScopy InChI
Affinity DataKi:  5.01nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419140(CHEMBL1830960)copy SMILEScopy InChI
Affinity DataKi:  6.31nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419135(CHEMBL1830962)copy SMILEScopy InChI
Affinity DataKi:  7.94nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419132(CHEMBL1830967)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419137(CHEMBL1830959)copy SMILEScopy InChI
Affinity DataKi:  19.9nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419132(CHEMBL1830967)copy SMILEScopy InChI
Affinity DataKi:  19.9nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419135(CHEMBL1830962)copy SMILEScopy InChI
Affinity DataKi:  19.9nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419139(CHEMBL1830966)copy SMILEScopy InChI
Affinity DataKi:  31.6nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419134(CHEMBL1830964)copy SMILEScopy InChI
Affinity DataKi:  31.6nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419134(CHEMBL1830964)copy SMILEScopy InChI
Affinity DataKi:  39.8nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419139(CHEMBL1830966)copy SMILEScopy InChI
Affinity DataKi:  50.1nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419130(CHEMBL1830956)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419140(CHEMBL1830960)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419138(CHEMBL1830957)copy SMILEScopy InChI
Affinity DataKi:  398nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419133(CHEMBL1830965)copy SMILEScopy InChI
Affinity DataKi:  501nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419130(CHEMBL1830956)copy SMILEScopy InChI
Affinity DataKi:  501nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419138(CHEMBL1830957)copy SMILEScopy InChI
Affinity DataKi:  631nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419133(CHEMBL1830965)copy SMILEScopy InChI
Affinity DataKi:  1.26E+3nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419141(CHEMBL1830958)copy SMILEScopy InChI
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre

Curated by ChEMBL
LigandPNGBDBM50419141(CHEMBL1830958)copy SMILEScopy InChI
Affinity DataKi: >3.16E+3nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4CGMPubMed