TargetOrexin receptor type 2(Rattus norvegicus (Rat))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.0776nMAssay Description:Antagonist activity at recombinant rat OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Rattus norvegicus (Rat))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.117nMAssay Description:Antagonist activity at recombinant rat OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.158nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.251nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.316nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.398nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.759nMAssay Description:Displacement of [3H]almorexant from recombinant human OX1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 0.794nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 1.29nMAssay Description:Displacement of [3H]almorexant from recombinant human OX2R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 5.01nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 5.01nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 6.31nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 7.94nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 19.9nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 19.9nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 19.9nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 31.6nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 31.6nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 50.1nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 398nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 501nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 501nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 1.26E+3nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Antagonist activity at recombinant human OX1R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
GlaxoSmithKline Medicine Research Centre
Curated by ChEMBL
Affinity DataKi: >3.16E+3nMAssay Description:Antagonist activity at recombinant human OX2R expressed in CHO cells by FLIPR calcium based functional assayMore data for this Ligand-Target Pair