TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Inhibitor constant was measured against Liver phosphorylase b in ratMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Inhibitor constant was measured against Muscle phosphorylase b in rabbitMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 5.10E+3nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 5.10E+3nMAssay Description:Inhibitor constant was measured against Muscle phosphorylase b in rabbitMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Inhibitor constant was measured against Liver phosphorylase b in ratMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 1.09E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase aMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 1.09E+4nMAssay Description:Inhibitor constant was measured against Muscle phosphorylase a in rabbitMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 1.28E+4nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 1.28E+4nMAssay Description:Inhibitor constant was measured against Liver phosphorylase b in ratMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 1.65E+4nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase aMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 1.65E+4nMAssay Description:Inhibitor constant was measured against Liver phosphorylase a in ratMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 1.65E+4nMAssay Description:Inhibitor constant was measured against Liver phosphorylase b in ratMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Inhibitor constant was measured against Muscle phosphorylase a in rabbitMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase aMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 2.98E+4nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase aMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Lajos Kossuth University
Curated by ChEMBL
Lajos Kossuth University
Curated by ChEMBL
Affinity DataKi: 2.98E+4nMAssay Description:Inhibitor constant was measured against Liver phosphorylase a in ratMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 3.10E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 3.20E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 8.10E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 1.05E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 1.05E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 1.44E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 3.70E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 4.40E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 7.10E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 1.70E+6nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 3.10E+6nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 7.40E+6nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 1.15E+7nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
PharmaHungary 2000 Kft.; TargetEx Kft.
US Patent
PharmaHungary 2000 Kft.; TargetEx Kft.
US Patent
Affinity DataIC50: 0.100nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
PharmaHungary 2000 Kft.; TargetEx Kft.
US Patent
PharmaHungary 2000 Kft.; TargetEx Kft.
US Patent
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.24E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.76E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.76E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMpH: 7.5 T: 2°CAssay Description:Stock solution of substrate (Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2) was prepared in DMSO at a concentration of 6 mM. Assays were performed in an as...More data for this Ligand-Target Pair
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