Affinity DataKi: 1.10nMAssay Description:Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.88E+3nMAssay Description:Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human CKIdeltaMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human CKIalphaMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human CKIalphaMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human CKIdeltaMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CK2More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CK2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.66E+5nMAssay Description:Inhibition of human JNK2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.75E+5nMAssay Description:Inhibition of human JNK1More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 3.85E+5nMAssay Description:Inhibition of human JNK1More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Istituto di Ricerche di Biologia Molecolare "P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 4.04E+5nMAssay Description:Inhibition of human JNK2More data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 143nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 146nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 393nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 522nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 124nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 498nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 46nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 202nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 929nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 897nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 92nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 708nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
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