TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Università degli Studi di Milano
Curated by ChEMBL
Università degli Studi di Milano
Curated by ChEMBL
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.95E+3nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Università degli Studi di Milano
Curated by ChEMBL
Università degli Studi di Milano
Curated by ChEMBL
Affinity DataIC50: 9.05E+3nMAssay Description:Inhibition of HDAC10More data for this Ligand-Target Pair
Affinity DataIC50: 1.77E+4nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Università degli Studi di Milano
Curated by ChEMBL
Università degli Studi di Milano
Curated by ChEMBL
Affinity DataIC50: 2.39E+4nMAssay Description:Inhibition of HDAC10More data for this Ligand-Target Pair
Affinity DataIC50: 2.67E+4nMAssay Description:Inhibition of HDAC3More data for this Ligand-Target Pair
Affinity DataIC50: 2.81E+4nMAssay Description:Inhibition of HDAC3More data for this Ligand-Target Pair
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of HDAC2More data for this Ligand-Target Pair