Compile Data Set for Download or QSAR
Found 151 with Last Name = 'walport' and Initial = 'l'
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395076(CHEMBL2164243)copy SMILEScopy InChI
Affinity DataKi:  1.97E+3nMAssay Description:Competitive inhibition of human KDM2A expressed in Escherichia coli using 2-oxoglutarate by enzyme kinetic assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395076(CHEMBL2164243)copy SMILEScopy InChI
Affinity DataKi:  8.50E+4nMAssay Description:Mixed type inhibition of human KDM2A expressed in Escherichia coli assessed inhibition constant for compound-enzyme-substrate complex using methyl ly...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395083(CHEMBL2164246)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human KDM4E expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50324535(3-{[9-(Dimethylamino)nonanoyl](hydroxy)amino}propa...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395083(CHEMBL2164246)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human KDM2A expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395078(CHEMBL2164245)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of human KDM2A expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50129197(4-(Hydroxyamino)-4-oxobutanoic acid | CHEMBL51979 ...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of human KDM4E expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50129197(4-(Hydroxyamino)-4-oxobutanoic acid | CHEMBL51979 ...)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of human KDM2A expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395083(CHEMBL2164246)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395083(CHEMBL2164246)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of human KDM5C catalytic domain expressed in Sf9 cells using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395076(CHEMBL2164243)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50197063(4,6-dioxoheptanoic acid | CHEMBL222824 | succinyla...)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of human KDM2A expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50324535(3-{[9-(Dimethylamino)nonanoyl](hydroxy)amino}propa...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of KDM4A (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 6B(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50129197(4-(Hydroxyamino)-4-oxobutanoic acid | CHEMBL51979 ...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human KDM6B catalytic domain expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395078(CHEMBL2164245)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human KDM5C catalytic domain expressed in Sf9 cells using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395076(CHEMBL2164243)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395076(CHEMBL2164243)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human KDM2A expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395076(CHEMBL2164243)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human KDM2A expressed in Escherichia coli by formaldehyde dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50129197(4-(Hydroxyamino)-4-oxobutanoic acid | CHEMBL51979 ...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50129197(4-(Hydroxyamino)-4-oxobutanoic acid | CHEMBL51979 ...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human KDM5C catalytic domain expressed in Sf9 cells using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395076(CHEMBL2164243)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human KDM7A catalytic domain expressed in Escherichia coli by MALDI assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50324535(3-{[9-(Dimethylamino)nonanoyl](hydroxy)amino}propa...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of KDM4C (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50197063(4,6-dioxoheptanoic acid | CHEMBL222824 | succinyla...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50440285(CHEMBL2424816)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395078(CHEMBL2164245)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395082(CHEMBL2164247)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human KDM2A expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)copy SMILEScopy InChI
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of KDM4A (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395078(CHEMBL2164245)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human KDM4E expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50197063(4,6-dioxoheptanoic acid | CHEMBL222824 | succinyla...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human KDM5C catalytic domain expressed in Sf9 cells using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395080(CHEMBL2164249)copy SMILEScopy InChI
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human PHD2 expressed in Escherichia coli by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50440289(CHEMBL2424812)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395080(CHEMBL2164249)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50440287(CHEMBL2424814)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50440292(CHEMBL2424809)copy SMILEScopy InChI
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM26113(2,4 PDCA | cid_10365 | pyridine carboxylate, 6a | ...)copy SMILEScopy InChI
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of KDM4C (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395080(CHEMBL2164249)copy SMILEScopy InChI
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human KDM2A expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50440290(CHEMBL2424811)copy SMILEScopy InChI
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395082(CHEMBL2164247)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50324535(3-{[9-(Dimethylamino)nonanoyl](hydroxy)amino}propa...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using H3K4me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395078(CHEMBL2164245)copy SMILEScopy InChI
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of human PHD2 expressed in Escherichia coli by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50440286(CHEMBL2424815)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50440288(CHEMBL2424813)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 6B(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50197063(4,6-dioxoheptanoic acid | CHEMBL222824 | succinyla...)copy SMILEScopy InChI
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of human KDM6B catalytic domain expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50129197(4-(Hydroxyamino)-4-oxobutanoic acid | CHEMBL51979 ...)copy SMILEScopy InChI
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of human PHD2 expressed in Escherichia coli by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50440285(CHEMBL2424816)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of KDM4C (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50197063(4,6-dioxoheptanoic acid | CHEMBL222824 | succinyla...)copy SMILEScopy InChI
Affinity DataIC50: 2.39E+4nMAssay Description:Inhibition of human KDM4E expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50440290(CHEMBL2424811)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of KDM4C (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50440288(CHEMBL2424813)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using H3K4me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395079(CHEMBL2164244)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
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