Compile Data Set for Download or QSAR
Found 464 with Last Name = 'westover' and Initial = 'l'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394718(CHEMBL2165801)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50161342(2-Amino-4-phenyl-indeno[1,2-d]pyrimidin-5-one | 2-...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317007(2-amino-4-(furan-2-yl)-5H-indeno[1,2-d]pyrimidin-5...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317008(2-amino-4-(5-chlorofuran-2-yl)-5H-indeno[1,2-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394722(CHEMBL2165807)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50317007(2-amino-4-(furan-2-yl)-5H-indeno[1,2-d]pyrimidin-5...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50394718(CHEMBL2165801)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50317008(2-amino-4-(5-chlorofuran-2-yl)-5H-indeno[1,2-d]pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317011(2-amino-4-(thiazol-2-yl)-5H-indeno[1,2-d]pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394717(CHEMBL2165802)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317010(2-amino-4-(thiophen-2-yl)-5H-indeno[1,2-d]pyrimidi...)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394719(CHEMBL2165800)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316892(2-amino-4-phenyl-8-(2-(pyridin-4-yl)ethylamino)-5H...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NXBPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316893(2-amino-4-phenyl-8-(2-(pyridin-2-yl)ethylamino)-5H...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NXBPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317003(2-amino-8-((morpholinoamino)methyl)-4-phenyl-5H-in...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50161342(2-Amino-4-phenyl-indeno[1,2-d]pyrimidin-5-one | 2-...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394720(CHEMBL2165799)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50491094(CHEMBL2377092)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Antagonist activity at human adenosine A2a receptor expressed in CHOK1 cells assessed as inhibition of NECA/forskolin-induced cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XPTPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394721(CHEMBL2165808)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394716(CHEMBL2165803)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317014(2-amino-4-(3-methoxyphenyl)-5H-indeno[1,2-d]pyrimi...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50394717(CHEMBL2165802)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394715(CHEMBL2165804)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50317003(2-amino-8-((morpholinoamino)methyl)-4-phenyl-5H-in...)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50394722(CHEMBL2165807)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50491101(CHEMBL2377103)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Antagonist activity at human adenosine A2a receptor expressed in CHOK1 cells assessed as inhibition of NECA/forskolin-induced cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XPTPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316992(2-amino-4-phenyl-9-(pyrrolidin-1-ylmethyl)-5H-inde...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50394719(CHEMBL2165800)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50317014(2-amino-4-(3-methoxyphenyl)-5H-indeno[1,2-d]pyrimi...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316899(2-amino-8-(4-methylpiperazin-1-yl)-4-phenyl-5H-ind...)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NXBPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316898(2-amino-8-morpholino-4-phenyl-5H-indeno[1,2-d]pyri...)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NXBPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50491105(CHEMBL2377110)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Antagonist activity at human adenosine A2a receptor expressed in CHOK1 cells assessed as inhibition of NECA/forskolin-induced cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XPTPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316997(2-amino-4-phenyl-8-((piperidin-1-ylamino)methyl)-5...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316895(2-Amino-8-[2-(1,1-dioxo-1lambda*6*-thiomorpholin-4...)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NXBPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50394723(CHEMBL2165806)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50317010(2-amino-4-(thiophen-2-yl)-5H-indeno[1,2-d]pyrimidi...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317022(2-amino-9-(morpholinomethyl)-4-phenyl-5H-indeno[1,...)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316993(2-amino-4-(4-fluorophenyl)-9-(pyrrolidin-1-ylmethy...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50491075(CHEMBL2377111)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Antagonist activity at human adenosine A2a receptor expressed in CHOK1 cells assessed as inhibition of NECA/forskolin-induced cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XPTPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317023(2-amino-4-(4-fluorophenyl)-9-(morpholinomethyl)-5H...)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317004(2-amino-4-phenyl-8-((pyrrolidin-1-ylamino)methyl)-...)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50330987(2-amino-4-phenyl-8-(pyrrolidin-1-ylmethyl)-5H-inde...)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at adenosine A2A receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1SCGPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50330987(2-amino-4-phenyl-8-(pyrrolidin-1-ylmethyl)-5H-inde...)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316894(2-amino-8-(2-morpholinoethylamino)-4-phenyl-5H-ind...)copy SMILEScopy InChI
Affinity DataKi:  4.40nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NXBPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50317012(2-amino-4-(pyridin-4-yl)-5H-indeno[1,2-d]pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50491100(CHEMBL2377228)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Antagonist activity at human adenosine A2a receptor expressed in CHOK1 cells assessed as inhibition of NECA/forskolin-induced cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XPTPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316891(2-amino-8-((2-(dimethylamino)ethyl)(methyl)amino)-...)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NXBPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316897(2-amino-8-((1-ethylpiperidin-4-yl)(methyl)amino)-4...)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NXBPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50394721(CHEMBL2165808)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ388QPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50316995(2-amino-8-((furan-2-ylmethylamino)methyl)-4-phenyl...)copy SMILEScopy InChI
Affinity DataKi:  5.30nMAssay Description:Antagonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB246HPubMed
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