Compile Data Set for Download or QSAR
Found 83 with Last Name = 'kennis' and Initial = 'le'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403738(CHEMBL351483)copy SMILEScopy InChI
Affinity DataIC50: 0.214nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403753(CHEMBL162682)copy SMILEScopy InChI
Affinity DataIC50: 0.240nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403755(CHEMBL163190)copy SMILEScopy InChI
Affinity DataIC50: 0.288nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403745(CHEMBL162490)copy SMILEScopy InChI
Affinity DataIC50: 0.295nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403748(CHEMBL162232)copy SMILEScopy InChI
Affinity DataIC50: 0.339nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403752(CHEMBL162370)copy SMILEScopy InChI
Affinity DataIC50: 0.347nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403740(CHEMBL165350)copy SMILEScopy InChI
Affinity DataIC50: 0.355nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403742(CHEMBL165796)copy SMILEScopy InChI
Affinity DataIC50: 0.447nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403744(LUSAPERIDONE)copy SMILEScopy InChI
Affinity DataIC50: 0.550nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403739(CHEMBL163247)copy SMILEScopy InChI
Affinity DataIC50: 0.589nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403750(CHEMBL351200)copy SMILEScopy InChI
Affinity DataIC50: 0.603nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403753(CHEMBL162682)copy SMILEScopy InChI
Affinity DataIC50: 0.617nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403747(CHEMBL162826)copy SMILEScopy InChI
Affinity DataIC50: 0.692nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403740(CHEMBL165350)copy SMILEScopy InChI
Affinity DataIC50: 0.692nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403745(CHEMBL162490)copy SMILEScopy InChI
Affinity DataIC50: 0.708nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403738(CHEMBL351483)copy SMILEScopy InChI
Affinity DataIC50: 0.724nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403748(CHEMBL162232)copy SMILEScopy InChI
Affinity DataIC50: 0.851nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403754(CHEMBL164612)copy SMILEScopy InChI
Affinity DataIC50: 0.891nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403738(CHEMBL351483)copy SMILEScopy InChI
Affinity DataIC50: 0.955nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403755(CHEMBL163190)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403746(CHEMBL162147)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403742(CHEMBL165796)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403752(CHEMBL162370)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403740(CHEMBL165350)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403739(CHEMBL163247)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403739(CHEMBL163247)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403750(CHEMBL351200)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403752(CHEMBL162370)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403755(CHEMBL163190)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403747(CHEMBL162826)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403744(LUSAPERIDONE)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403747(CHEMBL162826)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403749(CHEMBL165181)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403746(CHEMBL162147)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403745(CHEMBL162490)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403753(CHEMBL162682)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403750(CHEMBL351200)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403754(CHEMBL164612)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403751(CHEMBL162436)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403744(LUSAPERIDONE)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403748(CHEMBL162232)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403742(CHEMBL165796)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403751(CHEMBL162436)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403743(CHEMBL162058)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403746(CHEMBL162147)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403741(CHEMBL165677)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403751(CHEMBL162436)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403754(CHEMBL164612)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403737(CHEMBL165776)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)copy SMILEScopy InChI
Affinity DataIC50: 8.30nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72JMXPubMed
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