Compile Data Set for Download or QSAR
Found 69 with Last Name = 'prugar' and Initial = 'li'
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  541nMAssay Description:Binding affinity to biotinylated AAK1 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  1.75E+3nMAssay Description:Binding affinity to biotinylated GAK (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  4.40E+3nMAssay Description:Binding affinity to biotinylated BMP2K (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  1.19E+4nMAssay Description:Binding affinity to biotinylated STK16 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502299(CHEMBL4544854)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM311155((S)-N-(4-(4-((2-amino-4-methylpentyl)oxy)-3-cyanop...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM321107((S)-ethyl (8-((2-amino-2,4-dimethylpentyl)oxy)-6H-...)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM335593(3-((5-((4-aminopiperidin-1-yl)methyl)pyrrolo[2,1-f...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM279457((R)-1-(5-(7H-pyrrolo[2, 3-d]pyrimidin-4-yl)-1H-ben...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502295(CHEMBL4439128)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502283(CHEMBL4541962)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502285(CHEMBL4543869)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502308(CHEMBL4442812)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502304(CHEMBL4483684)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50445242(CHEMBL3102941)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502305(CHEMBL4443908)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502289(CHEMBL4444527)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502307(CHEMBL4454007)copy SMILEScopy InChI
Affinity DataIC50: 149nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502290(CHEMBL4524476)copy SMILEScopy InChI
Affinity DataIC50: 161nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502302(CHEMBL4474078)copy SMILEScopy InChI
Affinity DataIC50: 184nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502293(CHEMBL4461527)copy SMILEScopy InChI
Affinity DataIC50: 209nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502288(CHEMBL4561278)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50024286(CHEMBL3334981)copy SMILEScopy InChI
Affinity DataIC50: 319nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502297(CHEMBL4448513)copy SMILEScopy InChI
Affinity DataIC50: 381nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502291(CHEMBL4515873)copy SMILEScopy InChI
Affinity DataIC50: 381nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502300(CHEMBL4468845)copy SMILEScopy InChI
Affinity DataIC50: 387nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502306(CHEMBL4475520)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502296(CHEMBL4449852)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502284(CHEMBL4529052)copy SMILEScopy InChI
Affinity DataIC50: 462nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502292(CHEMBL4553067)copy SMILEScopy InChI
Affinity DataIC50: 612nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+3nMAssay Description:Binding affinity to biotinylated AAK1 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataIC50: 3.25E+3nMAssay Description:Binding affinity to biotinylated GAK (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502298(CHEMBL4471240)copy SMILEScopy InChI
Affinity DataIC50: 3.39E+3nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502294(CHEMBL4476807)copy SMILEScopy InChI
Affinity DataIC50: 4.44E+3nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataIC50: 1.01E+4nMAssay Description:Binding affinity to biotinylated BMP2K (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Binding affinity to biotinylated STK16 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataKd:  3.10nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502303(CHEMBL4455428)copy SMILEScopy InChI
Affinity DataKd:  53nMAssay Description:Binding affinity to wild type DNA-tagged human AAK1 (G25 to L333 residues) expressed in bacterial expression system by quantitative PCR based KINOMEs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288790(CHEMBL4167311)copy SMILEScopy InChI
Affinity DataKd:  7.20E+3nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288791(CHEMBL4162766)copy SMILEScopy InChI
Affinity DataKd:  1.60E+3nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288792(CHEMBL4163357)copy SMILEScopy InChI
Affinity DataKd:  19nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288793(CHEMBL4160425)copy SMILEScopy InChI
Affinity DataKd:  160nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50086268(CHEMBL3425867)copy SMILEScopy InChI
Affinity DataKd:  8.90nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288794(CHEMBL4166209)copy SMILEScopy InChI
Affinity DataKd:  970nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288795(CHEMBL4159403)copy SMILEScopy InChI
Affinity DataKd:  250nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288796(CHEMBL4168337)copy SMILEScopy InChI
Affinity DataKd:  210nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288797(CHEMBL4163801)copy SMILEScopy InChI
Affinity DataKd:  80nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288798(CHEMBL4171678)copy SMILEScopy InChI
Affinity DataKd:  52nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50086268(CHEMBL3425867)copy SMILEScopy InChI
Affinity DataKd:  4.5nMAssay Description:Inhibition of wild-type human partial length KIT (I571 to D952 residues) expressed in bacterial expression system by ATP-site competition binding ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DB9PubMed
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