Compile Data Set for Download or QSAR
Found 109 with Last Name = 'price' and Initial = 'lm'
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Inhibition of human norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
LigandPNGBDBM604244(US11661418, Compound I-15)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604251(Preparation of (2R,4S)—N—((S)-1-(((5-((Z)—N-hydrox...)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604250(Preparation of (2R,4S)-4-(3-(1H-pyrazol-1-yl)pheny...)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604249(Preparation of (2R,4S)—N—((S)-1-((4-carbamimidoylb...)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604246(Preparation of (S)—N-(4-carbamimidoylbenzyl)-1-((2...)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604240(Preparation of (2R,4S)—N—((S)-1-((4-((Z)—N′-...)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604241(Preparation of (2R,4S)-2-(((S)-1-((4-carbamimidoyl...)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604242(Preparation of ethyl 3-((2R,4S)-2-(((S)-1-((4-carb...)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604243(Preparation of 3-((2R,4S)-2-(((S)-1-((4-carbamimid...)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604245(US11661418, Compound I-16)copy SMILES
Affinity DataKi: <500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
TargetMacrophage metalloelastase(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi:  1.35E+3nMAssay Description:Inhibition of human MMP12More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
LigandPNGBDBM604247(Preparation of benzyl (imino(4-(((S)-1-((2R,4S)-4-...)copy SMILES
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604252(US11661418, Compound I-31)copy SMILES
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
LigandPNGBDBM604248(Preparation of benzyl ((4-(((S)-2-((2R,4S)-1-ethyl...)copy SMILES
Affinity DataKi:  6.25E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P2733R
TargetCollagenase 3(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi:  7.73E+3nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP14More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetStromelysin-2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP10More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrix metalloproteinase-15(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP15More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrix metalloproteinase-16(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP16More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrix metalloproteinase-20(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP20More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrix metalloproteinase-24(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP24More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrix metalloproteinase-25(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP25More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrix metalloproteinase-26(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP26More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetStromelysin-1(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetMatrilysin(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP7More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0H0WPubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50395921(CHEMBL2164511)copy SMILEScopy InChI
Affinity DataIC50: 0.511nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0VMVPubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485077(CHEMBL2023517)copy SMILEScopy InChI
Affinity DataIC50: 0.520nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485061(CHEMBL2023524)copy SMILEScopy InChI
Affinity DataIC50: 0.530nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50395911(CHEMBL2164521)copy SMILEScopy InChI
Affinity DataIC50: 0.657nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0VMVPubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50395920(CHEMBL2164512)copy SMILEScopy InChI
Affinity DataIC50: 0.850nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0VMVPubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50395910(CHEMBL2164522)copy SMILEScopy InChI
Affinity DataIC50: 0.912nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0VMVPubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485056(CHEMBL2023515)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485076(CHEMBL2023402)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485083(CHEMBL2023523)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485060(CHEMBL2023522)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485084(CHEMBL2023518)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50395909(CHEMBL2164523)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0VMVPubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485059(CHEMBL2023520)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485078(CHEMBL2023521)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485058(CHEMBL2023519)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50395908(CHEMBL2164524)copy SMILEScopy InChI
Affinity DataIC50: 1.39nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0VMVPubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50365344(CHEMBL1956115)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50485057(CHEMBL2023516)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W38050PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50395919(CHEMBL2164513)copy SMILEScopy InChI
Affinity DataIC50: 1.61nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0VMVPubMed
Displayed 1 to 50 (of 109 total ) | Next | Last >>
Jump to: