Compile Data Set for Download or QSAR
Found 28 with Last Name = 'rokosz' and Initial = 'lr'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223615(3-bromo-5-cyclohexyl-N-(pyridin-3-ylmethyl)pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223602(CHEMBL442802 | N-(2-(5-phenyl-7-(pyridin-3-ylmethy...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223587(3-bromo-5-(2-chlorophenyl)-N-((pyridin-3-yloxy)met...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223567(3-bromo-5-(2-chlorophenyl)-N-(pyridin-3-ylmethyl)p...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223590(3-bromo-5-(2-fluorophenyl)-N-((pyridin-3-yloxy)met...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223583(3-bromo-5-(piperidin-3-yl)-N-(pyridin-3-ylmethyl)p...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223580(3-bromo-5-(2-chlorophenyl)-N-methylpyrazolo[1,5-a]...)copy SMILEScopy InChI
Affinity DataIC50: 247nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223591(3-bromo-5-(furan-2-yl)-N-(pyridin-3-ylmethyl)pyraz...)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223578(3-bromo-5-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)p...)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223594(3-bromo-5-isopropyl-N-(pyridin-3-ylmethyl)pyrazolo...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223593(3-bromo-5-(2-chlorophenyl)-N-(4-(methylsulfonyl)ph...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223581(3-bromo-N-(pyridin-3-ylmethyl)-5-(thiophen-2-yl)py...)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223595(1-(3-bromo-7-(pyridin-3-ylmethylamino)pyrazolo[1,5...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223586(3-bromo-5-phenyl-N-(pyridin-3-ylmethyl)pyrazolo[1,...)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223609(3-bromo-5-phenyl-N-((pyridin-3-yloxy)methyl)pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223568(CHEMBL250183 | ethyl 3-bromo-7-(pyridin-3-ylmethyl...)copy SMILEScopy InChI
Affinity DataIC50: 790nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223608(3-bromo-5-ethyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5...)copy SMILEScopy InChI
Affinity DataIC50: 920nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223605(2-(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223573(3-bromo-5-cyclopropyl-N-(pyridin-3-ylmethyl)pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223577(3-bromo-5-(methylthio)-N-(pyridin-3-ylmethyl)pyraz...)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223601(3-bromo-5-methoxy-N-(pyridin-3-ylmethyl)pyrazolo[1...)copy SMILEScopy InChI
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223592(3-(methylthio)-5-phenyl-N-(pyridin-3-ylmethyl)pyra...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223607(3-ethyl-5-phenyl-N-(pyridin-3-ylmethyl)pyrazolo[1,...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223599(3-bromo-5-methyl-N-(pyridin-3-ylmethyl)pyrazolo[1,...)copy SMILEScopy InChI
Affinity DataIC50: 3.53E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223610(3-bromo-N5-methyl-N7-(pyridin-3-ylmethyl)pyrazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223576(3-ethynyl-5-phenyl-N-(pyridin-3-ylmethyl)pyrazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 9.82E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223570(3-bromo-5-(2-fluorophenyl)-N-phenylpyrazolo[1,5-a]...)copy SMILEScopy InChI
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50223582(CHEMBL249947 | N-benzyl-3-bromo-5-(2-fluorophenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07NDPubMed