Compile Data Set for Download or QSAR
Found 96 with Last Name = 'aoyagi-scharber' and Initial = 'm'
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50084621(BMN 673 | Talazoparib)copy SMILEScopy InChI
Affinity DataKi:  0.850nMAssay Description:Inhibition of human PARP2 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50084621(BMN 673 | Talazoparib)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50084621(BMN 673 | Talazoparib)copy SMILEScopy InChI
Affinity DataIC50: 0.570nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145154(CHEMBL3764920)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145152(CHEMBL3763446)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145151(CHEMBL3764202)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145135(CHEMBL3764188)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145138(CHEMBL3764085)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145092(CHEMBL3763531)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50446130(AG-014699 | AG-14447 | RUCAPARIB CAMSYLATE | Rucap...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145100(CHEMBL3765318)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145097(CHEMBL3764829)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145143(CHEMBL3765528)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145132(CHEMBL3765434)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145144(CHEMBL3764951)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145133(CHEMBL3763188)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145142(CHEMBL3765056)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145149(CHEMBL3763822)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145131(CHEMBL3765291)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145139(CHEMBL3765125)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145087(CHEMBL3764052)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145094(CHEMBL3764422)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145089(CHEMBL3764190)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145140(CHEMBL3763497)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145096(CHEMBL3765611)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145141(CHEMBL3764995)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145146(CHEMBL3763705)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145101(CHEMBL3763674)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145095(CHEMBL3764670)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145099(CHEMBL3763243)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145088(CHEMBL3765275)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145090(CHEMBL3764811)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145147(CHEMBL3765472)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145098(CHEMBL3763844)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145136(CHEMBL3763963)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145155(CHEMBL3765670)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145086(CHEMBL3764640)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145085(CHEMBL3763589)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145137(CHEMBL3763370)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145093(CHEMBL3763661)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145134(CHEMBL3764464)copy SMILEScopy InChI
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145145(CHEMBL3765661)copy SMILEScopy InChI
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50316226((S)-2-(4-(piperidin-3-yl)phenyl)-2H-indazole-7-car...)copy SMILEScopy InChI
Affinity DataIC50: 8.10nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145130(CHEMBL3765357)copy SMILEScopy InChI
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145091(CHEMBL3763164)copy SMILEScopy InChI
Affinity DataIC50: 9.60nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145104(CHEMBL3763348)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145150(CHEMBL3764066)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
BioMarin Pharmaceutical Inc.

Curated by ChEMBL
LigandPNGBDBM50145102(CHEMBL3764974)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of human PARP1 using [3H]NAD as substrate after 1 min by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35WJRPubMed
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