Compile Data Set for Download or QSAR
Found 86 with Last Name = 'arcuri' and Initial = 'm'
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109179(4-[3-(3-{3-[4-(3-Hydroxy-phenyl)-piperidin-1-yl]-p...)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109122(4-[3-(3-{3-[4-(3-Methoxy-phenyl)-piperidin-1-yl]-p...)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109188(4-[3-(3-{3-[4-(2-Methoxy-phenyl)-piperidin-1-yl]-p...)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429537(CHEMBL2333770)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429541(CHEMBL2333766)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429535(CHEMBL2333772)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429536(CHEMBL2333771)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109182(4-(3-{3-[3-(4-Cyclohexyl-piperidin-1-yl)-propyl]-u...)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109186(2,6-Dimethyl-4-(3-{3-[3-(4-phenyl-piperidin-1-yl)-...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109185(4-[3-(3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-p...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50060728((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429534(CHEMBL2333773)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429548(CHEMBL2333759)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429538(CHEMBL2333767)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429557(CHEMBL2333357)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429546(CHEMBL2333761)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429558(CHEMBL2333356)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429560(CHEMBL2333354)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429547(CHEMBL2333760)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109194(4-[3-(3-{3-[4-(3-Hydroxy-phenyl)-piperazin-1-yl]-p...)copy SMILEScopy InChI
Affinity DataKi:  37nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429567(CHEMBL2333776)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429561(CHEMBL2333353)copy SMILEScopy InChI
Affinity DataKi:  48nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109173(2,6-Dimethyl-4-(3-{3-[3-(4-phenyl-piperazin-1-yl)-...)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429562(CHEMBL2333352)copy SMILEScopy InChI
Affinity DataKi:  69nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429569(CHEMBL2333774)copy SMILEScopy InChI
Affinity DataKi:  75nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429545(CHEMBL2333762)copy SMILEScopy InChI
Affinity DataKi:  77nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429553(CHEMBL2333361)copy SMILEScopy InChI
Affinity DataKi:  84nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109193(4-(3-{3-[3-(4-Benzyl-piperidin-1-yl)-propyl]-ureid...)copy SMILEScopy InChI
Affinity DataKi:  84nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109178(2,6-Dimethyl-4-(3-{3-[3-(4-phenyl-piperidin-1-yl)-...)copy SMILEScopy InChI
Affinity DataKi:  89nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109183(2,6-Dimethyl-4-(3-{3-[3-(4-o-tolyl-piperazin-1-yl)...)copy SMILEScopy InChI
Affinity DataKi:  96nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109192(4-[3-(3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-p...)copy SMILEScopy InChI
Affinity DataKi:  105nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109180(4-[3-(3-{3-[4-(2-Hydroxy-phenyl)-piperazin-1-yl]-p...)copy SMILEScopy InChI
Affinity DataKi:  108nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429564(CHEMBL2333350)copy SMILEScopy InChI
Affinity DataKi:  128nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429563(CHEMBL2333351)copy SMILEScopy InChI
Affinity DataKi:  145nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429552(CHEMBL2333756)copy SMILEScopy InChI
Affinity DataKi:  169nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429568(CHEMBL2333775)copy SMILEScopy InChI
Affinity DataKi:  171nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429544(CHEMBL2333763)copy SMILEScopy InChI
Affinity DataKi:  172nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429540(CHEMBL2333768)copy SMILEScopy InChI
Affinity DataKi:  175nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109181(4-(3-{3-[3-(4-Biphenyl-3-yl-piperidin-1-yl)-propyl...)copy SMILEScopy InChI
Affinity DataKi:  188nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429559(CHEMBL2333355)copy SMILEScopy InChI
Affinity DataKi:  313nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109190(4-[3-(3-{3-[4-(4-Chloro-phenyl)-piperazin-1-yl]-pr...)copy SMILEScopy InChI
Affinity DataKi:  322nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109177(4-[3-(3-{3-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-p...)copy SMILEScopy InChI
Affinity DataKi:  405nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109184(2,6-Dimethyl-4-(3-{3-[3-(4-p-tolyl-piperazin-1-yl)...)copy SMILEScopy InChI
Affinity DataKi:  503nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429556(CHEMBL2333358)copy SMILEScopy InChI
Affinity DataKi:  506nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109176(2,6-Dimethyl-4-{3-[3-(3-piperidin-1-yl-propyl)-ure...)copy SMILEScopy InChI
Affinity DataKi:  523nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429555(CHEMBL2333359)copy SMILEScopy InChI
Affinity DataKi:  571nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429565(CHEMBL2333349)copy SMILEScopy InChI
Affinity DataKi:  607nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50429554(CHEMBL2333360)copy SMILEScopy InChI
Affinity DataKi:  644nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells assessed as residual [beta-33P] bound to plate after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R6GPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109189(4-[3-(3-{3-[4-(3,4-Dichloro-phenyl)-piperazin-1-yl...)copy SMILEScopy InChI
Affinity DataKi:  677nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109191(5-Cyano-4-[3-(3-{3-[4-(2-methoxy-phenyl)-piperazin...)copy SMILEScopy InChI
Affinity DataKi:  684nMAssay Description:Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DJ5DZ8PubMed
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