Compile Data Set for Download or QSAR
Found 86 with Last Name = 'awale' and Initial = 'm'
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50277545(4-(9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-benzo[...)copy SMILEScopy InChI
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50175305(CHEMBL3600873)copy SMILEScopy InChI
Affinity DataIC50: 0.0640nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50277545(4-(9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-benzo[...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50175305(CHEMBL3600873)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase B(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50277545(4-(9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-benzo[...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Aurora B kinase in human HeLa Kyoto cells assessed as effect on distribution of phspho-histone H3 ser10 level incubated for 20 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198027(CHEMBL3921246)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198027(CHEMBL3921246)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198081(CHEMBL3915550)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198080(CHEMBL3932394)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198082(CHEMBL3904239)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198086(CHEMBL3985313)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50277545(4-(9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-benzo[...)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Inhibition of Aurora A kinase autophosphorylation at Thr288 in human HeLa Kyoto cells incubated for 20 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase B(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50175305(CHEMBL3600873)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of Aurora B kinase in human HeLa Kyoto cells assessed as effect on distribution of phspho-histone H3 ser10 level incubated for 20 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198052(CHEMBL3896597)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of Aurora A kinase autophosphorylation at Thr288 in human HeLa Kyoto cells incubated for 20 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198052(CHEMBL3896597)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198044(CHEMBL3903187)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198045(CHEMBL3975102)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198027(CHEMBL3921246)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198079(CHEMBL3924918)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198078(CHEMBL3941377)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198084(CHEMBL3913242)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198077(CHEMBL3951166)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50175305(CHEMBL3600873)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of Aurora A kinase autophosphorylation at Thr288 in human HeLa Kyoto cells incubated for 20 hrsMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198076(CHEMBL3939478)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198042(CHEMBL3935395)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198041(CHEMBL3984254)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University of Berne

Curated by ChEMBL
LigandPNGBDBM96504(4-chloranyl-2-(2-naphthalen-1-yloxyethanoylamino)b...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9NCBPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198152(CHEMBL3923442)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198048(CHEMBL3941909)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198043(CHEMBL3983087)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198027(CHEMBL3921246)copy SMILEScopy InChI
Affinity DataIC50: 760nMAssay Description:Inhibition of Aurora A kinase autophosphorylation at Thr288 in human HeLa Kyoto cells incubated for 20 hrsMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198162(CHEMBL3938394)copy SMILEScopy InChI
Affinity DataIC50: 780nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198044(CHEMBL3903187)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198153(CHEMBL3924626)copy SMILEScopy InChI
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University of Berne

Curated by ChEMBL
LigandPNGBDBM50526037(CHEMBL4439848)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9NCBPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198027(CHEMBL3921246)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198086(CHEMBL3985313)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University of Berne

Curated by ChEMBL
LigandPNGBDBM50526038(CHEMBL4525597)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9NCBPubMed
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198082(CHEMBL3904239)copy SMILEScopy InChI
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University of Berne

Curated by ChEMBL
LigandPNGBDBM50526034(CHEMBL4540384)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9NCBPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198046(CHEMBL3911508)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198081(CHEMBL3915550)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198159(CHEMBL3956916)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198074(CHEMBL3914435)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198154(CHEMBL3949078)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198045(CHEMBL3975102)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198080(CHEMBL3932394)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of Aurora-B/INCENP (unknown origin) using biotinylated STK2 substrate incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University of Berne

Curated by ChEMBL
LigandPNGBDBM50526040(CHEMBL4447880)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9NCBPubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198049(CHEMBL3967949)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
TargetAurora kinase A(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50198157(CHEMBL3974813)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of His-tagged human Aurora A kinase (122 to 40 residues) expressed in Escherichia coli BL21 (DE3) Rosetta cells using biotinylated STK2 su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CM5PubMed
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