TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 151nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 510nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
Affinity DataKi: 730nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+3nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 1.71E+3nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 1.72E+3nMAssay Description:Inhibition human recombinant HcK using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 1.76E+3nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
Affinity DataKi: 1.86E+3nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£ degli Studi di Siena
Curated by ChEMBL
Universit£ degli Studi di Siena
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 2.16E+3nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£ degli Studi di Siena
Curated by ChEMBL
Universit£ degli Studi di Siena
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 2.81E+3nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 3.70E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 3.70E+3nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair