TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 156nMAssay Description:Inhibition of 5-HT uptake in rat synaptosomal fractionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 377nMAssay Description:Inhibition of noradrenaline uptake in rat synaptosomal fractionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human ERG by IonWorks patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human ERG by IonWorks patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human ERG by IonWorks patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human ERG by IonWorks patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human ERG by IonWorks patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£t D£sseldorf
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assayMore data for this Ligand-Target Pair
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